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99m-TC-PSMA-I&S

IRCCS San Raffaele · Phase 2 active Small molecule

99m-TC-PSMA-I&S is a radiopharmaceutical that targets prostate-specific membrane antigen (PSMA) for diagnostic imaging of prostate cancer.

99m-TC-PSMA-I&S is a radiopharmaceutical that targets prostate-specific membrane antigen (PSMA) for diagnostic imaging of prostate cancer. Used for Diagnostic imaging of prostate cancer.

At a glance

Generic name99m-TC-PSMA-I&S
SponsorIRCCS San Raffaele
Drug classRadiopharmaceutical
TargetPSMA
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 2

Mechanism of action

It works by binding to PSMA, a protein overexpressed on the surface of prostate cancer cells, allowing for visualization of tumors through positron emission tomography (PET) imaging. This enables accurate diagnosis and staging of prostate cancer, as well as assessment of treatment response.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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