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Incruse Ellipta — Competitive Intelligence Brief
marketed
Anticholinergic
Muscarinic acetylcholine receptor M4
Respiratory
Small molecule
Live · refreshed every 30 min
Target snapshot
Incruse Ellipta (UMECLIDINIUM) — Glaxo Grp England. Umeclidinium works by blocking the M4 muscarinic acetylcholine receptor to relax airway smooth muscle and improve breathing.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Incruse Ellipta TARGET | UMECLIDINIUM | Glaxo Grp England | marketed | Anticholinergic | Muscarinic acetylcholine receptor M4 | 2013-01-01 |
| Pentam | PENTAMIDINE | Fresenius Kabi | marketed | Antiprotozoal | Muscarinic acetylcholine receptor M4 | 1984-01-01 |
| Antrenyl | OXYPHENONIUM | Novartis | marketed | oxyphenonium | Muscarinic acetylcholine receptor M1, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M4 | 1982-01-01 |
| Methylrosaniline Chloride | GENTIAN VIOLET | marketed | Muscarinic acetylcholine receptor M4 | 1982-01-01 | ||
| Salagen | PILOCARPINE | marketed | Cholinergic Receptor Agonist | Muscarinic acetylcholine receptor M4 | 1974-01-01 | |
| Cephadol | DIPHENIDOL | marketed | Antiemetic | Muscarinic acetylcholine receptor M4 | 1967-01-01 | |
| Pro-Banthine | PROPANTHELINE | marketed | Anticholinergic | Muscarinic acetylcholine receptor M4 | 1953-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Anticholinergic class)
- · 4 drugs in this class
- Pearl Therapeutics, Inc. · 3 drugs in this class
- Shionogi · 2 drugs in this class
- Ain Shams University · 1 drug in this class
- Astellas Pharma Inc · 1 drug in this class
- Boehringer Ingelheim · 1 drug in this class
- Covis · 1 drug in this class
- Forest Labs Inc · 1 drug in this class
- Fougera Pharms · 1 drug in this class
- Glaxo Grp England · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Incruse Ellipta — Competitive Intelligence Brief. https://druglandscape.com/ci/umeclidinium. Accessed 2026-06-10.
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