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Tyrosine kinase inhibitor — Competitive Intelligence Brief

Tyrosine kinase inhibitor (Tyrosine kinase inhibitor) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Tyrosine kinase inhibitor. Area: Oncology.

phase 3 Tyrosine kinase inhibitor Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Tyrosine kinase inhibitor (Tyrosine kinase inhibitor) — Institut für Klinische Krebsforschung IKF GmbH at Krankenhaus Nordwest. Tyrosine kinase inhibitors block the activity of specific enzymes called tyrosine kinases, which are involved in the activation of proteins by signal transduction cascades.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Tyrosine kinase inhibitor TARGET Tyrosine kinase inhibitor Institut für Klinische Krebsforschung IKF GmbH at Krankenhaus Nordwest phase 3 Tyrosine kinase inhibitor
Inlyta Axitinib Pfizer marketed Receptor tyrosine kinase inhibitor Vascular endothelial growth factor receptors (VEGFR)-1, VEGFR-2, VEGFR-3 2012-01-01
DW6012(Dasidiem tab. 10/100mg) DW6012(Dasidiem tab. 10/100mg) Dong Wha Pharmaceutical Co. Ltd. marketed Tyrosine kinase inhibitor combination BCR-ABL, SRC family kinases
Dasatinib Tablets Dasatinib Tablets Chia Tai Tianqing Pharmaceutical Group Co., Ltd. marketed BCR-ABL tyrosine kinase inhibitor BCR-ABL, SRC family kinases
Cipterbin Combined With Vinorelbine Cipterbin Combined With Vinorelbine Zhejiang Cancer Hospital marketed Tyrosine kinase inhibitor combined with vinca alkaloid Multiple tyrosine kinases (cipterbin); tubulin (vinorelbine)
Anlotinib plus Pemetrexed Anlotinib plus Pemetrexed Henan Provincial People's Hospital marketed Multi-target tyrosine kinase inhibitor plus antifolate antimetabolite VEGFR, FGFR, RET, c-Kit (anlotinib); thymidylate synthase, DHFR, GARFT (pemetrexed)
Axitinib (AG-013736) axitinib-ag-013736 Pfizer marketed tyrosine kinase inhibitor vascular endothelial growth factor receptors (VEGFRs)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Tyrosine kinase inhibitor class)

  1. Jiangsu HengRui Medicine Co., Ltd. · 5 drugs in this class
  2. Centre Leon Berard · 2 drugs in this class
  3. AB Science · 2 drugs in this class
  4. Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 2 drugs in this class
  5. Betta Pharmaceuticals Co., Ltd. · 1 drug in this class
  6. Angion Biomedica Corp · 1 drug in this class
  7. Beijing InnoCare Pharma Tech Co., Ltd. · 1 drug in this class
  8. Chang-Ming Huang, Prof. · 1 drug in this class
  9. Deciphera Pharmaceuticals, LLC · 1 drug in this class
  10. AstraZeneca · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Tyrosine kinase inhibitor — Competitive Intelligence Brief. https://druglandscape.com/ci/tyrosine-kinase-inhibitor. Accessed 2026-05-16.

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