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Tukysa — Competitive Intelligence Brief
marketed
Kinase Inhibitor [EPC]
ERBB2/ERBB3
Oncology
Live · refreshed every 30 min
Target snapshot
Tukysa (tucatinib) — Seagen. Tukysa works by blocking the ERBB2/ERBB3 receptors, which are involved in the growth and spread of cancer cells.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Tukysa TARGET | tucatinib | Seagen | marketed | Kinase Inhibitor [EPC] | ERBB2/ERBB3 | 2020-01-01 |
| Tukysa | tukysa | Pfizer | marketed | Kinase Inhibitor [EPC] | ERBB2/ERBB3 | 2020-01-01 |
| Hernexeos | ZONGERTINIB | Boehringer Ingelheim | marketed | Kinase Inhibitor [EPC] | 2025-01-01 | |
| Wayrilz | RILZABRUTINIB | Genzyme Corp | marketed | Kinase Inhibitor [EPC] | 2025-01-01 | |
| Itovebi | INAVOLISIB | Genentech Inc | marketed | Kinase Inhibitor [EPC] | 2025-01-01 | |
| Romvimza | VIMSELTINIB | Deciphera Pharms | marketed | Kinase Inhibitor [EPC] | 2025-01-01 | |
| Itovebi | inavolisib | Pfizer | marketed | Kinase Inhibitor [EPC] | phosphatidylinositol 3-kinase (PI3K) alpha (PIK3CA) | 2024-01-01 |
Recent regulatory actions (last 90 days)
- — Hernexeos · FDA · approved · US · Boehringer Ingelheim
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Kinase Inhibitor [EPC] class)
- · 12 drugs in this class
- Pfizer · 7 drugs in this class
- Novartis · 3 drugs in this class
- Bayer · 2 drugs in this class
- Boehringer Ingelheim · 2 drugs in this class
- AstraZeneca · 2 drugs in this class
- Beigene Usa Inc · 1 drug in this class
- BeiGene · 1 drug in this class
- AbbVie · 1 drug in this class
- Bristol · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Tukysa — Competitive Intelligence Brief. https://druglandscape.com/ci/tucatinib. Accessed 2026-05-13.
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