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Trifluridine/Tipiracil + Regorafenib — Competitive Intelligence Brief

Trifluridine/Tipiracil + Regorafenib (Trifluridine/Tipiracil + Regorafenib) competitive landscape: 0 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Nucleoside analog + multikinase inhibitor combination. Area: Oncology.

phase 3 Nucleoside analog + multikinase inhibitor combination Thymidylate synthase (trifluridine/tipiracil); VEGFR, FGFR, KIT, RET, BRAF (regorafenib) Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Trifluridine/Tipiracil + Regorafenib (Trifluridine/Tipiracil + Regorafenib) — Second Affiliated Hospital, School of Medicine, Zhejiang University. This combination pairs a nucleoside analog that inhibits thymidylate synthase with a multikinase inhibitor targeting angiogenesis and tumor growth pathways.

Comparator set

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Trifluridine/Tipiracil + Regorafenib TARGET Trifluridine/Tipiracil + Regorafenib Second Affiliated Hospital, School of Medicine, Zhejiang University phase 3 Nucleoside analog + multikinase inhibitor combination Thymidylate synthase (trifluridine/tipiracil); VEGFR, FGFR, KIT, RET, BRAF (regorafenib)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Nucleoside analog + multikinase inhibitor combination class)

  1. Second Affiliated Hospital, School of Medicine, Zhejiang University · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Trifluridine/Tipiracil + Regorafenib — Competitive Intelligence Brief. https://druglandscape.com/ci/trifluridine-tipiracil-regorafenib. Accessed 2026-05-17.

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