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Trifluridine/Tipiracil + Regorafenib — Competitive Intelligence Brief
phase 3
Nucleoside analog + multikinase inhibitor combination
Thymidylate synthase (trifluridine/tipiracil); VEGFR, FGFR, KIT, RET, BRAF (regorafenib)
Oncology
Small molecule
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Target snapshot
Trifluridine/Tipiracil + Regorafenib (Trifluridine/Tipiracil + Regorafenib) — Second Affiliated Hospital, School of Medicine, Zhejiang University. This combination pairs a nucleoside analog that inhibits thymidylate synthase with a multikinase inhibitor targeting angiogenesis and tumor growth pathways.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Trifluridine/Tipiracil + Regorafenib TARGET | Trifluridine/Tipiracil + Regorafenib | Second Affiliated Hospital, School of Medicine, Zhejiang University | phase 3 | Nucleoside analog + multikinase inhibitor combination | Thymidylate synthase (trifluridine/tipiracil); VEGFR, FGFR, KIT, RET, BRAF (regorafenib) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Nucleoside analog + multikinase inhibitor combination class)
- Second Affiliated Hospital, School of Medicine, Zhejiang University · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Trifluridine/Tipiracil + Regorafenib — Competitive Intelligence Brief. https://druglandscape.com/ci/trifluridine-tipiracil-regorafenib. Accessed 2026-05-17.
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