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Trifluridine cures — Competitive Intelligence Brief

Trifluridine cures (Trifluridine cures) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Nucleoside analog; antimetabolite. Area: Oncology.

phase 3 Nucleoside analog; antimetabolite Thymidylate synthase; DNA Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Trifluridine cures (Trifluridine cures) — Centre Hospitalier Universitaire Dijon. Trifluridine is a nucleoside analog that inhibits thymidylate synthase and gets incorporated into DNA, disrupting cancer cell replication.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Trifluridine cures TARGET Trifluridine cures Centre Hospitalier Universitaire Dijon phase 3 Nucleoside analog; antimetabolite Thymidylate synthase; DNA
Suvemcitug injection, trifluridine/tipiracil tablets Suvemcitug injection, trifluridine/tipiracil tablets Jiangsu Simcere Pharmaceutical Co., Ltd. phase 3 Nucleoside analog; antimetabolite Thymidylate synthase; DNA
TS-1, oxaliplatin TS-1, oxaliplatin Samsung Medical Center phase 3 Fluoropyrimidine + platinum-based chemotherapy combination Thymidylate synthase; DNA (platinum crosslinking)
Fluoropyrimidine-based Chemotherapy Fluoropyrimidine-based Chemotherapy Hoffmann-La Roche phase 3 Antimetabolite chemotherapy Thymidylate synthase; DNA/RNA incorporation
Carac® (Fluorouracil) Cream Carac® (Fluorouracil) Cream Actavis Inc. phase 3 Antimetabolite; Pyrimidine analog Thymidylate synthase; DNA and RNA synthesis
CAPEOX/Capecitabine CAPEOX/Capecitabine Qilu Pharmaceutical Co., Ltd. phase 3 Antimetabolite; Fluoropyrimidine Thymidylate synthase; DNA/RNA synthesis
Pifeltro DORAVIRINE Merck & Co. marketed Human Immunodeficiency Virus 1 Non-Nucleoside Analog Reverse Transcriptase Inhibitor [EPC] 2018-01-01

Recent regulatory actions (last 90 days)

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Nucleoside analog; antimetabolite class)

  1. Assistance Publique - Hôpitaux de Paris · 1 drug in this class
  2. Astellas Pharma Global Development, Inc. · 1 drug in this class
  3. AstraZeneca · 1 drug in this class
  4. Celgene · 1 drug in this class
  5. Centre Hospitalier Universitaire Dijon · 1 drug in this class
  6. Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 1 drug in this class
  7. Chia Tai Tianqing Pharmaceutical Group Nanjing Shunxin Pharmaceutical Co., Ltd. · 1 drug in this class
  8. Eisai Inc. · 1 drug in this class
  9. Gruppo Italiano Malattie EMatologiche dell'Adulto · 1 drug in this class
  10. Jiangsu Simcere Pharmaceutical Co., Ltd. · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Trifluridine cures — Competitive Intelligence Brief. https://druglandscape.com/ci/trifluridine-cures. Accessed 2026-06-10.

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing