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Detrol — Competitive Intelligence Brief

Detrol (TOLTERODINE) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Cholinergic Muscarinic Antagonist. Area: Metabolic.

marketed Cholinergic Muscarinic Antagonist Muscarinic acetylcholine receptor M1 Metabolic Small molecule Live · refreshed every 30 min

Target snapshot

Detrol (TOLTERODINE) — Upjohn. Detrol works by blocking the action of a chemical called acetylcholine at the muscarinic receptors in the bladder muscle.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Detrol TARGET TOLTERODINE Upjohn marketed Cholinergic Muscarinic Antagonist Muscarinic acetylcholine receptor M1 1998-01-01
Northera DROXIDOPA Lundbeck Na Ltd marketed Catecholamine Muscarinic acetylcholine receptor M1 2014-01-01
Vesicare SOLIFENACIN Astellas Pharma marketed Cholinergic Muscarinic Antagonist Muscarinic acetylcholine receptor M1 2004-01-01
Evoxac CEVIMELINE Cosette marketed Cholinergic Receptor Agonist Muscarinic acetylcholine receptor M1 2000-01-01
Provocholine METHACHOLINE Methapharm marketed Cholinergic Receptor Agonist Muscarinic acetylcholine receptor M1 1986-01-01
Atrovent IPRATROPIUM marketed Anticholinergic Muscarinic acetylcholine receptor M1 1986-01-01
Carboxybenzylpenicillin CARBENICILLIN marketed Penicillin-class Antibacterial Muscarinic acetylcholine receptor M1 1982-01-01

Recent regulatory actions (last 90 days)

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Cholinergic Muscarinic Antagonist class)

  1. · 2 drugs in this class
  2. AbbVie · 2 drugs in this class
  3. Astellas Pharma · 1 drug in this class
  4. Hisamitsu Pharmaceutical Co., Inc. · 1 drug in this class
  5. Upjohn · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Detrol — Competitive Intelligence Brief. https://druglandscape.com/ci/tolterodine. Accessed 2026-05-14.

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