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Zelnorm — Competitive Intelligence Brief
marketed
Serotonin-4 Receptor Agonist
5-hydroxytryptamine receptor 2B
Metabolic
Small molecule
Live · refreshed every 30 min
Target snapshot
Zelnorm (TEGASEROD).
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Zelnorm TARGET | TEGASEROD | marketed | Serotonin-4 Receptor Agonist | 5-hydroxytryptamine receptor 2B | 2002-01-01 | |
| Mexitil | MEXILETINE | Boehringer Ingelheim | marketed | Antiarrhythmic | 5-hydroxytryptamine receptor 2B | 1985-01-01 |
| Forane | ISOFLURANE | Baxter | marketed | General Anesthetic [EPC] | 5-hydroxytryptamine receptor 2B | 1979-01-01 |
| Amoxil | amoxicillin | Generic (originally Beecham/GSK) | marketed | Aminopenicillin (Beta-lactam antibiotic) | 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2B, 5-hydroxytryptamine receptor 2C | 1972-01-01 |
| Nalidixate | NALIDIXIC ACID | marketed | nalidixic acid | 5-hydroxytryptamine receptor 2B | 1964-01-01 | |
| Cital | Cital | Ain Shams University | marketed | Solute carrier family 22 member 1, 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2B | ||
| Fenazoxine | NEFOPAM | marketed | nefopam | 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2B, 5-hydroxytryptamine receptor 2C |
Recent regulatory actions (last 90 days)
- — Mexitil · FDA · approved · US · Boehringer Ingelheim
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
- — Amoxil · 8778924 · Compound · US
- — Amoxil · 8357394 · Formulation · US
- — Amoxil · 8299052 · Method of Use · US
Sponsor landscape (Serotonin-4 Receptor Agonist class)
- · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Zelnorm — Competitive Intelligence Brief. https://druglandscape.com/ci/tegaserod. Accessed 2026-05-13.
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