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TAS-102, Regorafenib , Fruquintinib — Competitive Intelligence Brief
Target snapshot
TAS-102, Regorafenib , Fruquintinib (TAS-102, Regorafenib , Fruquintinib) — Suzhou Suncadia Biopharmaceuticals Co., Ltd.. TAS-102 is a nucleoside analog that inhibits thymidylate synthase, leading to DNA damage in cancer cells. Regorafenib is a multi-kinase inhibitor that targets angiogenic, stromal, and tumor cells. Fruquintinib is a potent and highly selective inhibitor of vascular endothelial growth factor receptor 2 (VEGFR2).
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| TAS-102, Regorafenib , Fruquintinib TARGET | TAS-102, Regorafenib , Fruquintinib | Suzhou Suncadia Biopharmaceuticals Co., Ltd. | phase 3 | Nucleoside analog, Multi-kinase inhibitor, VEGFR2 inhibitor | Thymidylate synthase, VEGFR2 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Nucleoside analog, Multi-kinase inhibitor, VEGFR2 inhibitor class)
- Suzhou Suncadia Biopharmaceuticals Co., Ltd. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). TAS-102, Regorafenib , Fruquintinib — Competitive Intelligence Brief. https://druglandscape.com/ci/tas-102-regorafenib-fruquintinib. Accessed 2026-05-17.
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