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TAS-102, Regorafenib , Fruquintinib — Competitive Intelligence Brief

TAS-102, Regorafenib , Fruquintinib (TAS-102, Regorafenib , Fruquintinib) competitive landscape: 0 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Nucleoside analog, Multi-kinase inhibitor, VEGFR2 inhibitor. Area: Oncology.

phase 3 Nucleoside analog, Multi-kinase inhibitor, VEGFR2 inhibitor Thymidylate synthase, VEGFR2 Oncology Small molecule Live · refreshed every 30 min

Target snapshot

TAS-102, Regorafenib , Fruquintinib (TAS-102, Regorafenib , Fruquintinib) — Suzhou Suncadia Biopharmaceuticals Co., Ltd.. TAS-102 is a nucleoside analog that inhibits thymidylate synthase, leading to DNA damage in cancer cells. Regorafenib is a multi-kinase inhibitor that targets angiogenic, stromal, and tumor cells. Fruquintinib is a potent and highly selective inhibitor of vascular endothelial growth factor receptor 2 (VEGFR2).

Comparator set

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
TAS-102, Regorafenib , Fruquintinib TARGET TAS-102, Regorafenib , Fruquintinib Suzhou Suncadia Biopharmaceuticals Co., Ltd. phase 3 Nucleoside analog, Multi-kinase inhibitor, VEGFR2 inhibitor Thymidylate synthase, VEGFR2

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Nucleoside analog, Multi-kinase inhibitor, VEGFR2 inhibitor class)

  1. Suzhou Suncadia Biopharmaceuticals Co., Ltd. · 1 drug in this class

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Cite this brief

Drug Landscape (2026). TAS-102, Regorafenib , Fruquintinib — Competitive Intelligence Brief. https://druglandscape.com/ci/tas-102-regorafenib-fruquintinib. Accessed 2026-05-17.

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