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Tamoxifen + Aminoglutethimide — Competitive Intelligence Brief
phase 3
SERM and CYP11A1 inhibitor
estrogen receptor
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Tamoxifen + Aminoglutethimide (Tamoxifen + Aminoglutethimide) — Austrian Breast & Colorectal Cancer Study Group. Tamoxifen acts as a selective estrogen receptor modulator (SERM) to inhibit estrogen's action in breast tissue, while aminoglutethimide inhibits the enzyme CYP11A1, which is involved in the synthesis of steroids, including estrogen.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Tamoxifen + Aminoglutethimide TARGET | Tamoxifen + Aminoglutethimide | Austrian Breast & Colorectal Cancer Study Group | phase 3 | SERM and CYP11A1 inhibitor | estrogen receptor | |
| Orserdu | ELACESTRANT | Stemline Therap | marketed | Estrogen Receptor Antagonist [EPC] | Estrogen receptor | 2023-01-01 |
| Nextstellis | ESTETROL | Mayne Pharma | marketed | Estrogen | Estrogen receptor | 2021-01-01 |
| Cerianna | FLUOROESTRADIOL F-18 | GE HealthCare | marketed | Radioactive Diagnostic Agent [EPC] | Estrogen receptor | 2020-01-01 |
| Duavee | conjugated-estrogens-bazedoxifene | Pfizer | marketed | Estrogen [EPC] | estrogen receptors α and β | 2013-01-01 |
| Osphena | OSPEMIFENE | Duchesnay | marketed | Estrogen Agonist/Antagonist [EPC] | Estrogen receptor beta | 2013-01-01 |
| Duavee | BAZEDOXIFENE | Wyeth Pharms Pfizer | marketed | Estrogen [EPC] | estrogen receptors (ER) α and β | 2013-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
- — Duavee · 7683051 · US
Sponsor landscape (SERM and CYP11A1 inhibitor class)
- Austrian Breast & Colorectal Cancer Study Group · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Tamoxifen + Aminoglutethimide — Competitive Intelligence Brief. https://druglandscape.com/ci/tamoxifen-aminoglutethimide. Accessed 2026-05-16.
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