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Rocuronium bolus maintenance — Competitive Intelligence Brief
phase 3
Non-depolarizing neuromuscular blocker
Nicotinic acetylcholine receptor
Anesthesiology
Small molecule
Live · refreshed every 30 min
Target snapshot
Rocuronium bolus maintenance (Rocuronium bolus maintenance) — Merck Sharp & Dohme LLC. Rocuronium acts as a competitive antagonist at the nicotinic acetylcholine receptor, preventing acetylcholine from binding and thereby inhibiting muscle contraction.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Rocuronium bolus maintenance TARGET | Rocuronium bolus maintenance | Merck Sharp & Dohme LLC | phase 3 | Non-depolarizing neuromuscular blocker | Nicotinic acetylcholine receptor | |
| Succinylcholine Chloride | SUXAMETHONIUM | Novartis | marketed | Depolarizing Neuromuscular Blocker | Muscle-type nicotinic acetylcholine receptor | 1952-01-01 |
| nicotine nasal spray | nicotine nasal spray | Heinrich-Heine University, Duesseldorf | marketed | Nicotinic receptor agonist | Nicotinic acetylcholine receptors | |
| Succinylcholine + Neostigmine | Succinylcholine + Neostigmine | Brno University Hospital | marketed | Neuromuscular blocking agent reversal combination | Nicotinic acetylcholine receptor; acetylcholinesterase | |
| Galantamine-CR | Galantamine-CR | Massachusetts General Hospital | marketed | Cholinesterase inhibitor with nicotinic receptor allosteric modulator | Acetylcholinesterase; nicotinic acetylcholine receptors | |
| Rocuronium or Vecuronium | Rocuronium or Vecuronium | Merck Sharp & Dohme LLC | marketed | Neuromuscular blocking agent (non-depolarizing) | Nicotinic acetylcholine receptor at the neuromuscular junction | |
| Nicotine gum (C) | Nicotine gum (C) | 22nd Century Group, Inc. | marketed | Nicotinic acetylcholine receptor agonist | Nicotinic acetylcholine receptors |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Non-depolarizing neuromuscular blocker class)
- Merck Sharp & Dohme LLC · 2 drugs in this class
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Cite this brief
Drug Landscape (2026). Rocuronium bolus maintenance — Competitive Intelligence Brief. https://druglandscape.com/ci/rocuronium-bolus-maintenance. Accessed 2026-06-10.
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