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Rimegepant 75mg daily dosing — Competitive Intelligence Brief
marketed
calcitonin gene-related peptide receptor antagonist
calcitonin gene-related peptide receptor
Neuroscience
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Target snapshot
Rimegepant 75mg daily dosing (rimegepant-75mg-daily-dosing) — Pfizer. Rimegepant is a calcitonin gene-related peptide receptor antagonist that inhibits the release of pro-inflammatory peptides.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Rimegepant 75mg daily dosing TARGET | rimegepant-75mg-daily-dosing | Pfizer | marketed | calcitonin gene-related peptide receptor antagonist | calcitonin gene-related peptide receptor | |
| Nurtec Odt | rimegepant | Pfizer | marketed | Calcitonin Gene-related Peptide Receptor Antagonist | calcitonin gene-related peptide receptor | 2020-01-01 |
| Rimegepant/BHV3000 | rimegepant-bhv3000 | Pfizer | marketed | pharmacological class not specified | calcitonin gene-related peptide receptor (CGRPR) | |
| Rimegepant 75mg every other day dosing | rimegepant-75mg-every-other-day-dosing | Pfizer | marketed | calcitonin gene-related peptide receptor antagonist | calcitonin gene-related peptide receptor | |
| Rimegepant for acute migraine treatment | rimegepant-for-acute-migraine-treatment | Pfizer | marketed | calcitonin gene-related peptide receptor antagonist | calcitonin gene-related peptide receptor | |
| Rimegepant 75mg Orally Disintegrating Tablets (ODT) | rimegepant-75mg-orally-disintegrating-tablets-odt | Pfizer | marketed | calcitonin gene-related peptide receptor antagonist | calcitonin gene-related peptide receptor | |
| Zavegepant 100mg immediate release tablet | zavegepant-100mg-immediate-release-tablet | Pfizer Inc. | marketed | calcitonin gene-related peptide receptor antagonist | calcitonin gene-related peptide receptor (CGRPR) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (calcitonin gene-related peptide receptor antagonist class)
- Pfizer · 5 drugs in this class
- Pfizer Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Rimegepant 75mg daily dosing — Competitive Intelligence Brief. https://druglandscape.com/ci/rimegepant-75mg-daily-dosing. Accessed 2026-05-17.
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