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Rescue medications for sacituzumab tirumotecan — Competitive Intelligence Brief

Rescue medications for sacituzumab tirumotecan (Rescue medications for sacituzumab tirumotecan) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: antibody-drug conjugate. Area: Oncology.

phase 3 antibody-drug conjugate Trop-2 Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Rescue medications for sacituzumab tirumotecan (Rescue medications for sacituzumab tirumotecan) — Merck Sharp & Dohme LLC. Sacituzumab govitecan is an antibody-drug conjugate that targets Trop-2, delivering a cytotoxic payload to cancer cells.

Comparator set (6 drugs)

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DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Rescue medications for sacituzumab tirumotecan TARGET Rescue medications for sacituzumab tirumotecan Merck Sharp & Dohme LLC phase 3 antibody-drug conjugate Trop-2
Sacituzumab Govitecan (SG) Sacituzumab Govitecan (SG) University of California, Irvine phase 3 Antibody-drug conjugate (ADC) Trop-2 (TACSTD2)
Dato-DXd Dato-DXd AstraZeneca phase 3 Antibody-drug conjugate (ADC) TROP-2 (Trophoblast cell surface antigen 2)
DS-1062a DS-1062a Gustave Roussy, Cancer Campus, Grand Paris phase 3 Antibody-drug conjugate (ADC) TROP-2 (Trophoblast cell surface antigen 2)
Tisotumab Vedotin tivdak SEAGEN marketed Antibody-Drug Conjugate (ADC) Tissue factor 2021-01-01
LONCASTUXIMAB TESIRINE LONCASTUXIMAB TESIRINE marketed Antibody-Drug Conjugate (ADC) CD19 2021-01-01
Tivdak tisotumab-vedotin SEAGEN marketed Antibody-drug conjugate Tissue factor 2021-01-01

Recent regulatory actions (last 90 days)

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (antibody-drug conjugate class)

  1. Merck Sharp & Dohme LLC · 1 drug in this class
  2. Pfizer · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Rescue medications for sacituzumab tirumotecan — Competitive Intelligence Brief. https://druglandscape.com/ci/rescue-medications-for-sacituzumab-tirumotecan. Accessed 2026-05-17.

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