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Relugolix Combination Tablet — Competitive Intelligence Brief

Relugolix Combination Tablet (Relugolix Combination Tablet) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: GnRH receptor antagonist. Area: Oncology.

phase 3 GnRH receptor antagonist GnRH receptor Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Relugolix Combination Tablet (Relugolix Combination Tablet) — Sumitomo Pharma Switzerland GmbH. Relugolix combination tablet works by inhibiting gonadotropin-releasing hormone (GnRH) receptors, leading to a decrease in luteinizing hormone (LH) and follicle-stimulating hormone (FSH) production, which in turn reduces testosterone levels.

Comparator set (6 drugs)

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DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Relugolix Combination Tablet TARGET Relugolix Combination Tablet Sumitomo Pharma Switzerland GmbH phase 3 GnRH receptor antagonist GnRH receptor
Lupron leuprorelin Accord Healthcare S.L.U. marketed Gonadotropin Releasing Hormone Receptor Agonist GnRH receptors 1985-01-01
Micronor norethisterone Johnson & Johnson marketed Progestin GnRH receptors 1962-01-01
LHRHa LHRHa Imperial College London marketed LHRH agonist LHRH receptor (GnRH receptor)
GnRH agonist/antagonist GnRH agonist/antagonist Memorial Sloan Kettering Cancer Center marketed GnRH agonist/antagonist GnRH receptor
Cetrorelix and Leuprolide Cetrorelix and Leuprolide Instituto Valenciano de Infertilidad, IVI VALENCIA marketed GnRH antagonist and GnRH agonist combination GnRH receptor
Half-Dose Depot Triptorelin Half-Dose Depot Triptorelin Tehran University of Medical Sciences marketed GnRH agonist GnRH receptor

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

Sponsor landscape (GnRH receptor antagonist class)

  1. Sumitomo Pharma Switzerland GmbH · 1 drug in this class
  2. University of Michigan · 1 drug in this class
  3. VA Office of Research and Development · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Relugolix Combination Tablet — Competitive Intelligence Brief. https://druglandscape.com/ci/relugolix-combination-tablet. Accessed 2026-05-14.

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