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Relugolix Combination Tablet — Competitive Intelligence Brief
phase 3
GnRH receptor antagonist
GnRH receptor
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Relugolix Combination Tablet (Relugolix Combination Tablet) — Sumitomo Pharma Switzerland GmbH. Relugolix combination tablet works by inhibiting gonadotropin-releasing hormone (GnRH) receptors, leading to a decrease in luteinizing hormone (LH) and follicle-stimulating hormone (FSH) production, which in turn reduces testosterone levels.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Relugolix Combination Tablet TARGET | Relugolix Combination Tablet | Sumitomo Pharma Switzerland GmbH | phase 3 | GnRH receptor antagonist | GnRH receptor | |
| Lupron | leuprorelin | Accord Healthcare S.L.U. | marketed | Gonadotropin Releasing Hormone Receptor Agonist | GnRH receptors | 1985-01-01 |
| Micronor | norethisterone | Johnson & Johnson | marketed | Progestin | GnRH receptors | 1962-01-01 |
| LHRHa | LHRHa | Imperial College London | marketed | LHRH agonist | LHRH receptor (GnRH receptor) | |
| GnRH agonist/antagonist | GnRH agonist/antagonist | Memorial Sloan Kettering Cancer Center | marketed | GnRH agonist/antagonist | GnRH receptor | |
| Cetrorelix and Leuprolide | Cetrorelix and Leuprolide | Instituto Valenciano de Infertilidad, IVI VALENCIA | marketed | GnRH antagonist and GnRH agonist combination | GnRH receptor | |
| Half-Dose Depot Triptorelin | Half-Dose Depot Triptorelin | Tehran University of Medical Sciences | marketed | GnRH agonist | GnRH receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (GnRH receptor antagonist class)
- Sumitomo Pharma Switzerland GmbH · 1 drug in this class
- University of Michigan · 1 drug in this class
- VA Office of Research and Development · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Relugolix Combination Tablet — Competitive Intelligence Brief. https://druglandscape.com/ci/relugolix-combination-tablet. Accessed 2026-05-14.
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