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Regorafenib (BAY73-4506) — Competitive Intelligence Brief
phase 3
Multikinase inhibitor
VEGFR1-3, FGFR, TIE2, KIT, RET, RAF-1, BRAF
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Regorafenib (BAY73-4506) (Regorafenib (BAY73-4506)) — Bayer. Regorafenib is a multikinase inhibitor that blocks multiple receptor tyrosine kinases involved in tumor angiogenesis, stromal signaling, and oncogenic signaling.
Comparator set (1 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Regorafenib (BAY73-4506) TARGET | Regorafenib (BAY73-4506) | Bayer | phase 3 | Multikinase inhibitor | VEGFR1-3, FGFR, TIE2, KIT, RET, RAF-1, BRAF | |
| Trifluridine/Tipiracil + Regorafenib | Trifluridine/Tipiracil + Regorafenib | Second Affiliated Hospital, School of Medicine, Zhejiang University | phase 3 | Nucleoside analog + multikinase inhibitor combination | Thymidylate synthase (trifluridine/tipiracil); VEGFR, FGFR, KIT, RET, BRAF (regorafenib) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Multikinase inhibitor class)
- Bayer · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Regorafenib (BAY73-4506) — Competitive Intelligence Brief. https://druglandscape.com/ci/regorafenib-bay73-4506. Accessed 2026-05-16.
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