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Placebo to Tolterodine — Competitive Intelligence Brief
phase 3
Muscarinic M3 receptor antagonist
M3 muscarinic acetylcholine receptor
Urology
Small molecule
Live · refreshed every 30 min
Target snapshot
Placebo to Tolterodine (Placebo to Tolterodine) — Astellas Pharma Inc. Tolterodine is a muscarinic M3 receptor antagonist that reduces bladder muscle contractions to treat overactive bladder symptoms.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Placebo to Tolterodine TARGET | Placebo to Tolterodine | Astellas Pharma Inc | phase 3 | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| Solifenacin for 24 weeks | Solifenacin for 24 weeks | National Taiwan University Hospital | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| Toviaz (Fesoterodine) | Toviaz (Fesoterodine) | Weill Medical College of Cornell University | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| Spiriva HandiHaler | Spiriva HandiHaler | Chia Tai Tianqing Pharmaceutical Group Co., Ltd. | marketed | Long-acting muscarinic antagonist (LAMA) | M3 muscarinic acetylcholine receptor | |
| Solifenacin succinate treatment | Solifenacin succinate treatment | Barrie Urology Associates | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| Solifenacin PO | Solifenacin PO | Seattle Urology Research Center | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| Drug: ipratropium (AtroventTM) | Drug: ipratropium (AtroventTM) | AstraZeneca | marketed | Anticholinergic bronchodilator | M3 muscarinic acetylcholine receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Muscarinic M3 receptor antagonist class)
- Astellas Pharma Inc · 2 drugs in this class
- Barrie Urology Associates · 1 drug in this class
- National Taiwan University Hospital · 1 drug in this class
- Pfizer · 1 drug in this class
- Seattle Urology Research Center · 1 drug in this class
- Weill Medical College of Cornell University · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Placebo to Tolterodine — Competitive Intelligence Brief. https://druglandscape.com/ci/placebo-to-tolterodine. Accessed 2026-05-17.
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