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oxaliplatin plus capecitabine — Competitive Intelligence Brief
marketed
Platinum-based chemotherapy combination
DNA (oxaliplatin); thymidylate synthase (capecitabine/5-FU)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
oxaliplatin plus capecitabine (oxaliplatin plus capecitabine) — LiNing. Oxaliplatin and capecitabine work together as a chemotherapy combination where oxaliplatin cross-links DNA to prevent replication while capecitabine is converted to fluorouracil to inhibit thymidylate synthase and disrupt nucleotide synthesis.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| oxaliplatin plus capecitabine TARGET | oxaliplatin plus capecitabine | LiNing | marketed | Platinum-based chemotherapy combination | DNA (oxaliplatin); thymidylate synthase (capecitabine/5-FU) | |
| Oxaliplatin;Capecitabine | Oxaliplatin;Capecitabine | Hebei Medical University | marketed | Platinum-based chemotherapy combination; antimetabolite | DNA (oxaliplatin); thymidylate synthase (capecitabine/5-FU) | |
| atezolizumab + avastin + platinum-based chemotherapy | atezolizumab + avastin + platinum-based chemotherapy | ARCAGY/ GINECO GROUP | phase 3 | PD-L1 inhibitor + VEGF inhibitor + platinum-based chemotherapy combination | PD-L1, VEGF, DNA (platinum adducts) | |
| TS-1, oxaliplatin | TS-1, oxaliplatin | Samsung Medical Center | phase 3 | Fluoropyrimidine + platinum-based chemotherapy combination | Thymidylate synthase; DNA (platinum crosslinking) | |
| Oxaliplatin, calcium folinate, 5-fluorouracil | Oxaliplatin, calcium folinate, 5-fluorouracil | Karolinska University Hospital | phase 3 | Platinum-based chemotherapy combination (FOLFOX regimen) | DNA (oxaliplatin); thymidylate synthase (5-fluorouracil) | |
| Capecitabine & Oxaliplatin | Capecitabine & Oxaliplatin | Samsung Medical Center | phase 3 | Antimetabolite and platinum-based chemotherapy combination | Thymidylate synthase (capecitabine/5-FU); DNA (oxaliplatin) | |
| Pemetrexed+carboplatin/Cisplatin | Pemetrexed+carboplatin/Cisplatin | Suzhou Puhe Pharmaceutical Technology Co., LTD | phase 3 | Antifolate antimetabolite + platinum-based chemotherapy combination | Thymidylate synthase, dihydrofolate reductase, glycinamide ribonucleotide formyltransferase; DNA (platinum agents) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Platinum-based chemotherapy combination class)
- LiNing · 1 drug in this class
- Suzhou Suncadia Biopharmaceuticals Co., Ltd. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). oxaliplatin plus capecitabine — Competitive Intelligence Brief. https://druglandscape.com/ci/oxaliplatin-plus-capecitabine. Accessed 2026-05-16.
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