Last reviewed · How we verify
overencapsulated caffeine — Competitive Intelligence Brief
phase 3
stimulant
adenosine receptor
Central Nervous System
Small molecule
Live · refreshed every 30 min
Target snapshot
overencapsulated caffeine (overencapsulated caffeine) — Astellas Pharma Inc. Overencapsulated caffeine acts as a stimulant by increasing the levels of dopamine and norepinephrine in the brain.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| overencapsulated caffeine TARGET | overencapsulated caffeine | Astellas Pharma Inc | phase 3 | stimulant | adenosine receptor | |
| Nourianz | ISTRADEFYLLINE | Kyowa Kirin | marketed | CYP3A4 Substrates | Adenosine receptor A2a | 2019-01-01 |
| Singulair | montelukast | Merck & Co. | marketed | Leukotriene receptor antagonist (LTRA) | Cytochrome P450 2C8, Adenosine receptor A3, Cysteinyl leukotriene receptor 2 | 1998-02-20 |
| Neurontin | gabapentin | Generic (originally Parke-Davis/Pfizer) | marketed | Gabapentinoid (anticonvulsant/neuropathic pain agent) | Large neutral amino acids transporter small subunit 1, Adenosine receptor A1, Alpha-2A adrenergic receptor | 1993-12-30 |
| Lariam | MEFLOQUINE HYDROCHLORIDE | marketed | Antimalarial | Adenosine receptor A2a | 1989-01-01 | |
| Adenocard | ADENOSINE | Astellas Pharma | marketed | Adenosine Receptor Agonist [EPC] | Adenosine receptor A3 | 1989-01-01 |
| Lariam | MEFLOQUINE | marketed | Antimalarial | Adenosine receptor A2a | 1989-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (stimulant class)
- Astellas Pharma Inc · 1 drug in this class
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Cite this brief
Drug Landscape (2026). overencapsulated caffeine — Competitive Intelligence Brief. https://druglandscape.com/ci/overencapsulated-caffeine. Accessed 2026-06-10.
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