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overencapsulated caffeine — Competitive Intelligence Brief

overencapsulated caffeine (overencapsulated caffeine) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: stimulant. Area: Central Nervous System.

phase 3 stimulant adenosine receptor Central Nervous System Small molecule Live · refreshed every 30 min

Target snapshot

overencapsulated caffeine (overencapsulated caffeine) — Astellas Pharma Inc. Overencapsulated caffeine acts as a stimulant by increasing the levels of dopamine and norepinephrine in the brain.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
overencapsulated caffeine TARGET overencapsulated caffeine Astellas Pharma Inc phase 3 stimulant adenosine receptor
Nourianz ISTRADEFYLLINE Kyowa Kirin marketed CYP3A4 Substrates Adenosine receptor A2a 2019-01-01
Singulair montelukast Merck & Co. marketed Leukotriene receptor antagonist (LTRA) Cytochrome P450 2C8, Adenosine receptor A3, Cysteinyl leukotriene receptor 2 1998-02-20
Neurontin gabapentin Generic (originally Parke-Davis/Pfizer) marketed Gabapentinoid (anticonvulsant/neuropathic pain agent) Large neutral amino acids transporter small subunit 1, Adenosine receptor A1, Alpha-2A adrenergic receptor 1993-12-30
Lariam MEFLOQUINE HYDROCHLORIDE marketed Antimalarial Adenosine receptor A2a 1989-01-01
Adenocard ADENOSINE Astellas Pharma marketed Adenosine Receptor Agonist [EPC] Adenosine receptor A3 1989-01-01
Lariam MEFLOQUINE marketed Antimalarial Adenosine receptor A2a 1989-01-01

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (stimulant class)

  1. Astellas Pharma Inc · 1 drug in this class

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Cite this brief

Drug Landscape (2026). overencapsulated caffeine — Competitive Intelligence Brief. https://druglandscape.com/ci/overencapsulated-caffeine. Accessed 2026-06-10.

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