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O6-benzylguanine — Competitive Intelligence Brief
phase 3
DNA repair inhibitor / Alkyltransferase inhibitor
O6-alkylguanine-DNA alkyltransferase (AGT)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
O6-benzylguanine (O6-benzylguanine) — Case Comprehensive Cancer Center. O6-benzylguanine is an alkyltransferase inhibitor that depletes the DNA repair protein O6-alkylguanine-DNA alkyltransferase (AGT), sensitizing cancer cells to alkylating chemotherapy agents.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| O6-benzylguanine TARGET | O6-benzylguanine | Case Comprehensive Cancer Center | phase 3 | DNA repair inhibitor / Alkyltransferase inhibitor | O6-alkylguanine-DNA alkyltransferase (AGT) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (DNA repair inhibitor / Alkyltransferase inhibitor class)
- Case Comprehensive Cancer Center · 1 drug in this class
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Cite this brief
Drug Landscape (2026). O6-benzylguanine — Competitive Intelligence Brief. https://druglandscape.com/ci/o6-benzylguanine. Accessed 2026-05-17.
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