Last reviewed · How we verify
Niacin plus laropiprant — Competitive Intelligence Brief
marketed
Lipid-modifying agent combination
DP1 receptor (laropiprant component); niacin acts on GPR109A and other pathways
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Niacin plus laropiprant (Niacin plus laropiprant) — Institut Investigacio Sanitaria Pere Virgili. Niacin raises HDL cholesterol and lowers triglycerides, while laropiprant blocks prostaglandin D2 receptors to reduce niacin-induced flushing.
Comparator set (1 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Niacin plus laropiprant TARGET | Niacin plus laropiprant | Institut Investigacio Sanitaria Pere Virgili | marketed | Lipid-modifying agent combination | DP1 receptor (laropiprant component); niacin acts on GPR109A and other pathways | |
| Comparator: niacin + laropiprant | Comparator: niacin + laropiprant | Merck Sharp & Dohme LLC | phase 3 | Lipid-modifying agent combination | Niacin: GPR109A (hydroxycarboxylic acid receptor 2); Laropiprant: DP1 (prostaglandin D2 receptor) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Lipid-modifying agent combination class)
- Institut Investigacio Sanitaria Pere Virgili · 1 drug in this class
- Merck Sharp & Dohme LLC · 1 drug in this class
Subscribe to ongoing alerts
Push every new event for this competitive set into your RSS reader, IFTTT/Zapier workflow, or email digest:
- Niacin plus laropiprant CI watch — RSS
- Niacin plus laropiprant CI watch — Atom
- Niacin plus laropiprant CI watch — JSON
- Niacin plus laropiprant alone — RSS
- Whole Lipid-modifying agent combination class — RSS
Cite this brief
Drug Landscape (2026). Niacin plus laropiprant — Competitive Intelligence Brief. https://druglandscape.com/ci/niacin-plus-laropiprant. Accessed 2026-06-10.
Build your own brief
Pick any drug + add comparators:
https://druglandscape.com/ci/{slug}— auto-detected competitorshttps://druglandscape.com/ci/{slug}?vs=drug1,drug2,drug3— explicit comparators- Brand names auto-resolve:
/ci/keytruda→ 301 →/ci/pembrolizumab
Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing