Last reviewed · How we verify
Naltrexone plus Gabapentin — Competitive Intelligence Brief
phase 3
Opioid antagonist + anticonvulsant/analgesic combination
Opioid receptors (mu, delta, kappa) + voltage-gated calcium channels (Cav2.1, Cav2.2)
Psychiatry/Addiction Medicine
Small molecule
Live · refreshed every 30 min
Target snapshot
Naltrexone plus Gabapentin (Naltrexone plus Gabapentin) — Medical University of South Carolina. Naltrexone blocks opioid receptors while gabapentin modulates calcium channels and GABA neurotransmission to reduce pain and cravings in opioid use disorder.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Naltrexone plus Gabapentin TARGET | Naltrexone plus Gabapentin | Medical University of South Carolina | phase 3 | Opioid antagonist + anticonvulsant/analgesic combination | Opioid receptors (mu, delta, kappa) + voltage-gated calcium channels (Cav2.1, Cav2.2) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Opioid antagonist + anticonvulsant/analgesic combination class)
- Medical University of South Carolina · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Naltrexone plus Gabapentin — Competitive Intelligence Brief. https://druglandscape.com/ci/naltrexone-plus-gabapentin. Accessed 2026-05-15.
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