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néfopam — Competitive Intelligence Brief
marketed
Non-opioid analgesic; monoamine reuptake inhibitor
Norepinephrine transporter (NET); dopamine transporter (DAT); serotonin transporter (SERT)
Pain Management
Small molecule
Live · refreshed every 30 min
Target snapshot
néfopam (néfopam) — University Hospital, Bordeaux. Nefopam is a non-opioid analgesic that inhibits the reuptake of monoamines (norepinephrine, dopamine, and serotonin) in the central nervous system to produce analgesia.
Comparator set (5 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| néfopam TARGET | néfopam | University Hospital, Bordeaux | marketed | Non-opioid analgesic; monoamine reuptake inhibitor | Norepinephrine transporter (NET); dopamine transporter (DAT); serotonin transporter (SERT) | |
| Nefopam administration and prelevment | Nefopam administration and prelevment | University Hospital, Rouen | marketed | Non-opioid analgesic; monoamine reuptake inhibitor | Norepinephrine transporter, dopamine transporter, serotonin transporter | |
| Tesomet "Low dose" in fasted condition | Tesomet "Low dose" in fasted condition | Saniona | marketed | Monoamine reuptake inhibitor + biguanide combination | Serotonin transporter (SERT), norepinephrine transporter (NET), dopamine transporter (DAT); metformin targets mitochondrial glycerophosphate dehydrogenase | |
| Tesomet "High dose" in fed condition | Tesomet "High dose" in fed condition | Saniona | marketed | Monoamine reuptake inhibitor + biguanide combination | Serotonin transporter (SERT), norepinephrine transporter (NET), dopamine transporter (DAT); metformin targets mitochondrial glycerophosphate dehydrogenase | |
| Centanafadine SR | Centanafadine SR | Otsuka Pharmaceutical Development & Commercialization, Inc. | phase 3 | Triple monoamine reuptake inhibitor | Serotonin transporter (SERT), norepinephrine transporter (NET), dopamine transporter (DAT) | |
| Nefopam ampule | Nefopam ampule | Ministry Of Health / Nineveh Health Directorate | phase 3 | Non-opioid analgesic; monoamine reuptake inhibitor | Norepinephrine transporter, dopamine transporter, serotonin transporter |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Non-opioid analgesic; monoamine reuptake inhibitor class)
- Ministry Of Health / Nineveh Health Directorate · 1 drug in this class
- University Hospital, Bordeaux · 1 drug in this class
- University Hospital, Rouen · 1 drug in this class
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Cite this brief
Drug Landscape (2026). néfopam — Competitive Intelligence Brief. https://druglandscape.com/ci/n-fopam. Accessed 2026-05-16.
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