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metformin+ gliclazide — Competitive Intelligence Brief
marketed
Antidiabetic combination (biguanide + sulfonylurea)
Metformin: mitochondrial glycerophosphate dehydrogenase; Gliclazide: ATP-sensitive potassium channels on pancreatic beta cells
Diabetes
Small molecule
Live · refreshed every 30 min
Target snapshot
metformin+ gliclazide (metformin+ gliclazide) — GlaxoSmithKline. This combination reduces blood glucose by increasing insulin secretion and improving insulin sensitivity in type 2 diabetes patients.
Comparator set (2 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| metformin+ gliclazide TARGET | metformin+ gliclazide | GlaxoSmithKline | marketed | Antidiabetic combination (biguanide + sulfonylurea) | Metformin: mitochondrial glycerophosphate dehydrogenase; Gliclazide: ATP-sensitive potassium channels on pancreatic beta cells | |
| metformin + glimepiride | metformin + glimepiride | GlaxoSmithKline | marketed | Antidiabetic combination (biguanide + sulfonylurea) | Metformin: mitochondrial glycerophosphate dehydrogenase; Glimepiride: ATP-sensitive potassium channel (KATP) | |
| MET + Glibenclamide Group | MET + Glibenclamide Group | Hospital de Clinicas de Porto Alegre | marketed | Antidiabetic combination (biguanide + sulfonylurea) | AMPK pathway (metformin); ATP-sensitive potassium channel (glibenclamide) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Antidiabetic combination (biguanide + sulfonylurea) class)
- GlaxoSmithKline · 2 drugs in this class
- Hospital de Clinicas de Porto Alegre · 1 drug in this class
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Cite this brief
Drug Landscape (2026). metformin+ gliclazide — Competitive Intelligence Brief. https://druglandscape.com/ci/metformin-gliclazide. Accessed 2026-05-16.
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