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Low dose pilocarpine — Competitive Intelligence Brief
phase 3
Muscarinic receptor agonist
Muscarinic acetylcholine receptors (M3, M4)
Ophthalmology
Small molecule
Live · refreshed every 30 min
Target snapshot
Low dose pilocarpine (Low dose pilocarpine) — Ocuphire Pharma, Inc.. Low-dose pilocarpine is a muscarinic acetylcholine receptor agonist that stimulates parasympathetic activity to increase aqueous humor outflow and reduce intraocular pressure.
Comparator set (4 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Low dose pilocarpine TARGET | Low dose pilocarpine | Ocuphire Pharma, Inc. | phase 3 | Muscarinic receptor agonist | Muscarinic acetylcholine receptors (M3, M4) | |
| Pilocarpine Ophthalmic Solution | Pilocarpine Ophthalmic Solution | Maastricht University Medical Center | marketed | Muscarinic receptor agonist | Muscarinic acetylcholine receptor (M3) | |
| Pilocarpine HCl | Pilocarpine HCl | Allergan | phase 3 | Muscarinic receptor agonist | Muscarinic M3 receptor | |
| Xanomeline Enteric Capsule | Xanomeline Enteric Capsule | Bristol-Myers Squibb | phase 3 | muscarinic receptor agonist | M1, M4 | |
| Aceclidine ophthalmic solution | Aceclidine ophthalmic solution | LENZ Therapeutics, Inc | phase 3 | Muscarinic receptor agonist | Muscarinic acetylcholine receptors (M1, M3) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Muscarinic receptor agonist class)
- Allergan · 1 drug in this class
- LENZ Therapeutics, Inc · 1 drug in this class
- Maastricht University Medical Center · 1 drug in this class
- Ocuphire Pharma, Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Low dose pilocarpine — Competitive Intelligence Brief. https://druglandscape.com/ci/low-dose-pilocarpine. Accessed 2026-06-10.
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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing