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lithium plus valproate — Competitive Intelligence Brief
marketed
Mood stabilizer combination
GSK-3, inositol monophosphatase, histone deacetylase, GABA signaling
Psychiatry
Small molecule
Live · refreshed every 30 min
Target snapshot
lithium plus valproate (lithium plus valproate) — University of Sao Paulo. Lithium and valproate together modulate neuronal signaling and gene expression through distinct pathways to stabilize mood and reduce manic or depressive episodes.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| lithium plus valproate TARGET | lithium plus valproate | University of Sao Paulo | marketed | Mood stabilizer combination | GSK-3, inositol monophosphatase, histone deacetylase, GABA signaling | |
| Risperidone, divalproex | Risperidone, divalproex | Nathan Kline Institute for Psychiatric Research | marketed | Atypical antipsychotic + anticonvulsant mood stabilizer combination | Dopamine D2 receptor (risperidone); histone deacetylase / GABA pathway (divalproex) | |
| Quetiapine and Topiramate | Quetiapine and Topiramate | University of Cincinnati | marketed | Atypical antipsychotic + anticonvulsant mood stabilizer combination | D2 dopamine receptor, 5-HT2A serotonin receptor (quetiapine); voltage-gated sodium channels, carbonic anhydrase (topiramate) | |
| sodium valproate with Clozapine | sodium valproate with Clozapine | Shanghai Mental Health Center | marketed | Antipsychotic + mood stabilizer combination | Dopamine D2 receptor, serotonin 5-HT2A receptor, GABA pathways, histone deacetylase | |
| lithium plus carbamazepine | lithium plus carbamazepine | University of Sao Paulo | marketed | Mood stabilizer combination | Lithium: inositol monophosphatase and GSK-3β; Carbamazepine: voltage-gated sodium channels | |
| Paroxetine+Lamotrigine | Paroxetine+Lamotrigine | Ministry of Health & Welfare, Korea | marketed | SSRI + anticonvulsant mood stabilizer combination | Serotonin transporter (SERT); voltage-gated sodium channels; glutamate release modulation | |
| Paroxetine+Lithium | Paroxetine+Lithium | Ministry of Health & Welfare, Korea | marketed | SSRI + mood stabilizer combination | Serotonin transporter (SERT); inositol monophosphatase; protein kinase C |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Mood stabilizer combination class)
- University of Sao Paulo · 2 drugs in this class
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Cite this brief
Drug Landscape (2026). lithium plus valproate — Competitive Intelligence Brief. https://druglandscape.com/ci/lithium-plus-valproate. Accessed 2026-05-14.
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