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lisaftoclax +BTK inhibitor — Competitive Intelligence Brief
phase 3
BCL-2 inhibitor + BTK inhibitor combination
BCL-2 and BTK (Bruton's tyrosine kinase)
Oncology
Small molecule
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Target snapshot
lisaftoclax +BTK inhibitor (lisaftoclax +BTK inhibitor) — Ascentage Pharma Group Inc.. Lisaftoclax is a BCL-2 inhibitor combined with a BTK inhibitor to promote apoptosis in cancer cells while blocking B-cell survival signaling.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| lisaftoclax +BTK inhibitor TARGET | lisaftoclax +BTK inhibitor | Ascentage Pharma Group Inc. | phase 3 | BCL-2 inhibitor + BTK inhibitor combination | BCL-2 and BTK (Bruton's tyrosine kinase) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (BCL-2 inhibitor + BTK inhibitor combination class)
- Ascentage Pharma Group Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). lisaftoclax +BTK inhibitor — Competitive Intelligence Brief. https://druglandscape.com/ci/lisaftoclax-btk-inhibitor. Accessed 2026-05-18.
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