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Upstene — Competitive Intelligence Brief
marketed
Sodium-dependent serotonin transporter
Other
Small molecule
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Target snapshot
Upstene (INDALPINE).
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Upstene TARGET | INDALPINE | marketed | Sodium-dependent serotonin transporter | |||
| Fetzima | LEVOMILNACIPRAN | AbbVie | marketed | Serotonin and Norepinephrine Reuptake Inhibitor | Sodium-dependent serotonin transporter | 2013-01-01 |
| Pristiq | desvenlafaxine | Alembic Pharms Ltd | marketed | Serotonin and Norepinephrine Reuptake Inhibitor | Sodium-dependent serotonin transporter | 2008-01-01 |
| Celexa | CITALOPRAM | AbbVie | marketed | Serotonin Reuptake Inhibitor | Sodium-dependent serotonin transporter | 1998-01-01 |
| Plavix | clopidogrel | Generic (originally Sanofi/BMS) | marketed | Thienopyridine antiplatelet agent | Cytochrome P450 2B6, P2Y purinoceptor 12, Sodium-dependent serotonin transporter | 1997-11-17 |
| Racemic Sibutramine | SIBUTRAMINE | marketed | Norepinephrine, Serotonin, and Dopamine Reuptake Inhibitor Anorectic | Sodium-dependent serotonin transporter | 1997-01-01 | |
| Serzone | NEFAZODONE | Bristol-Myers Squibb | marketed | Serotonin Reuptake Inhibitor | Sodium-dependent serotonin transporter | 1994-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape
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Cite this brief
Drug Landscape (2026). Upstene — Competitive Intelligence Brief. https://druglandscape.com/ci/indalpine. Accessed 2026-05-13.
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