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Imipenem/Cilastatin/Relebactam — Competitive Intelligence Brief
marketed
Carbapenem antibiotic with beta-lactamase inhibitor
Bacterial penicillin-binding proteins; serine beta-lactamases
Infectious Disease
Small molecule
Live · refreshed every 30 min
Target snapshot
Imipenem/Cilastatin/Relebactam (Imipenem/Cilastatin/Relebactam) — Evopoint Biosciences Inc.. Imipenem/cilastatin/relebactam is a combination of a broad-spectrum beta-lactam antibiotic, a renal dehydropeptidase inhibitor, and a beta-lactamase inhibitor that together kill bacteria by inhibiting cell wall synthesis while protecting against enzymatic degradation.
Comparator set (1 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Imipenem/Cilastatin/Relebactam TARGET | Imipenem/Cilastatin/Relebactam | Evopoint Biosciences Inc. | marketed | Carbapenem antibiotic with beta-lactamase inhibitor | Bacterial penicillin-binding proteins; serine beta-lactamases | |
| Imipenem, Cilastatin and Relebactam | Imipenem, Cilastatin and Relebactam | Joseph L. Kuti, PharmD | marketed | Carbapenem antibiotic with beta-lactamase inhibitor | Penicillin-binding proteins (PBPs); beta-lactamase inhibition |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Carbapenem antibiotic with beta-lactamase inhibitor class)
- Evopoint Biosciences Inc. · 1 drug in this class
- Joseph L. Kuti, PharmD · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Imipenem/Cilastatin/Relebactam — Competitive Intelligence Brief. https://druglandscape.com/ci/imipenem-cilastatin-relebactam. Accessed 2026-05-18.
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