Last reviewed · How we verify
iloprost (5 µg) — Competitive Intelligence Brief
phase 3
prostacyclin analogue
prostacyclin receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
iloprost (5 µg) (iloprost (5 µg)) — Actelion. Iloprost is a prostacyclin analogue that acts as a vasodilator and inhibits platelet aggregation.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| iloprost (5 µg) TARGET | iloprost (5 µg) | Actelion | phase 3 | prostacyclin analogue | prostacyclin receptor | |
| Uptravi | SELEXIPAG | AstraZeneca | marketed | Prostacyclin Receptor Agonist [EPC] | Prostacyclin receptor | 2015-01-01 |
| Remodulin | TREPROSTINIL | United Therap | marketed | Prostacycline Vasodilator [EPC] | Prostacyclin receptor | 2002-01-01 |
| Flolan | EPOPROSTENOL | AstraZeneca | marketed | Prostacycline Vasodilator [EPC] | Prostacyclin receptor | 1995-01-01 |
| Fundyl | ENPROSTIL | marketed | enprostil | Prostacyclin receptor, Prostaglandin E2 receptor EP1 subtype, Prostaglandin E2 receptor EP3 subtype | ||
| FLOLAN injection with reformulated diluent | FLOLAN injection with reformulated diluent | GlaxoSmithKline | marketed | Prostacyclin analog | Prostacyclin receptor (IP receptor) | |
| prostacyclin | prostacyclin | United Therapeutics | marketed | P2Y purinoceptor 12, Prostacyclin receptor, Prostaglandin E2 receptor EP1 subtype |
Recent regulatory actions (last 90 days)
- — Uptravi · FDA · approved · US · AstraZeneca
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (prostacyclin analogue class)
- Actelion · 1 drug in this class
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Cite this brief
Drug Landscape (2026). iloprost (5 µg) — Competitive Intelligence Brief. https://druglandscape.com/ci/iloprost-5-g. Accessed 2026-06-10.
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