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High dose Oliceridine — Competitive Intelligence Brief
marketed
Mu-opioid receptor agonist (biased agonist)
Mu-opioid receptor (OPRM1)
Pain Management
Small molecule
Live · refreshed every 30 min
Target snapshot
High dose Oliceridine (High dose Oliceridine) — Nanjing First Hospital, Nanjing Medical University. Oliceridine is a mu-opioid receptor agonist that selectively activates G-protein signaling pathways to provide analgesia with potentially reduced beta-arrestin signaling.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| High dose Oliceridine TARGET | High dose Oliceridine | Nanjing First Hospital, Nanjing Medical University | marketed | Mu-opioid receptor agonist (biased agonist) | Mu-opioid receptor (OPRM1) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Mu-opioid receptor agonist (biased agonist) class)
- Nanjing First Hospital, Nanjing Medical University · 1 drug in this class
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Cite this brief
Drug Landscape (2026). High dose Oliceridine — Competitive Intelligence Brief. https://druglandscape.com/ci/high-dose-oliceridine. Accessed 2026-06-10.
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