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GSK 573719 +GW642444 125/25 — Competitive Intelligence Brief
phase 3
Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA)
Muscarinic M3 receptor; Beta-2 adrenergic receptor
Respiratory / Pulmonology
Small molecule
Live · refreshed every 30 min
Target snapshot
GSK 573719 +GW642444 125/25 (GSK 573719 +GW642444 125/25) — GlaxoSmithKline. This combination inhaler delivers a long-acting muscarinic antagonist (umeclidinium) and a long-acting beta-2 agonist (vilanterol) to relax airway smooth muscle and improve airflow in chronic obstructive pulmonary disease.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| GSK 573719 +GW642444 125/25 TARGET | GSK 573719 +GW642444 125/25 | GlaxoSmithKline | phase 3 | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; Beta-2 adrenergic receptor | |
| Tiotropium & olodaterol | Tiotropium & olodaterol | University of Dundee | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| UMEC/VI | UMEC/VI | GlaxoSmithKline | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| GSK573719/VI 62.5/25 | GSK573719/VI 62.5/25 | GlaxoSmithKline | phase 3 | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| Glycopyrronium/Formoterol Fumarate | Glycopyrronium/Formoterol Fumarate | AstraZeneca | phase 3 | LAMA/LABA combination (Long-Acting Muscarinic Antagonist / Long-Acting Beta-2 Agonist) | Muscarinic M3 receptor; Beta-2 adrenergic receptor | |
| Umeclidinium/Vilanterol 62.5/25 mcgs | Umeclidinium/Vilanterol 62.5/25 mcgs | National Institute of Respiratory Diseases, Mexico | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | M3 muscarinic receptor; beta-2 adrenergic receptor | |
| Aclidinium bromide & formoterol fumarate | Aclidinium bromide & formoterol fumarate | University of Dundee | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | M3 muscarinic receptor; beta-2 adrenergic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) class)
- GlaxoSmithKline · 5 drugs in this class
- University of Dundee · 2 drugs in this class
- National Institute of Respiratory Diseases, Mexico · 1 drug in this class
- University of Tennessee Graduate School of Medicine · 1 drug in this class
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Cite this brief
Drug Landscape (2026). GSK 573719 +GW642444 125/25 — Competitive Intelligence Brief. https://druglandscape.com/ci/gsk-573719-gw642444-125-25. Accessed 2026-05-18.
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