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Glycopyrronium/Formoterol Fumarate — Competitive Intelligence Brief
phase 3
LAMA/LABA combination (Long-Acting Muscarinic Antagonist / Long-Acting Beta-2 Agonist)
Muscarinic M3 receptor; Beta-2 adrenergic receptor
Respiratory / Pulmonology
Small molecule
Live · refreshed every 30 min
Target snapshot
Glycopyrronium/Formoterol Fumarate (Glycopyrronium/Formoterol Fumarate) — AstraZeneca. Glycopyrronium is an anticholinergic agent that blocks muscarinic receptors to reduce airway secretions and improve bronchial tone, while formoterol is a long-acting beta-2 agonist that relaxes airway smooth muscle to improve airflow.
Comparator set (4 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Glycopyrronium/Formoterol Fumarate TARGET | Glycopyrronium/Formoterol Fumarate | AstraZeneca | phase 3 | LAMA/LABA combination (Long-Acting Muscarinic Antagonist / Long-Acting Beta-2 Agonist) | Muscarinic M3 receptor; Beta-2 adrenergic receptor | |
| Tiotropium & olodaterol | Tiotropium & olodaterol | University of Dundee | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| UMEC/VI | UMEC/VI | GlaxoSmithKline | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| GSK573719/VI 62.5/25 | GSK573719/VI 62.5/25 | GlaxoSmithKline | phase 3 | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| GSK 573719 +GW642444 125/25 | GSK 573719 +GW642444 125/25 | GlaxoSmithKline | phase 3 | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; Beta-2 adrenergic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (LAMA/LABA combination (Long-Acting Muscarinic Antagonist / Long-Acting Beta-2 Agonist) class)
- AstraZeneca · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Glycopyrronium/Formoterol Fumarate — Competitive Intelligence Brief. https://druglandscape.com/ci/glycopyrronium-formoterol-fumarate. Accessed 2026-05-18.
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