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Gimeracil and Oteracil Porassium Capsules — Competitive Intelligence Brief
phase 2
Pyrimidine synthesis inhibitor
Dihydroorotate dehydrogenase
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Gimeracil and Oteracil Porassium Capsules (Gimeracil and Oteracil Porassium Capsules) — Beijing Biohealthcare Biotechnology Co.,Ltd. Inhibits dihydroorotate dehydrogenase
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Gimeracil and Oteracil Porassium Capsules TARGET | Gimeracil and Oteracil Porassium Capsules | Beijing Biohealthcare Biotechnology Co.,Ltd | phase 2 | Pyrimidine synthesis inhibitor | Dihydroorotate dehydrogenase | |
| Aubagio | TERIFLUNOMIDE | Sanofi | marketed | Pyrimidine Synthesis Inhibitor [EPC] | dihydroorotate dehydrogenase | 2012-01-01 |
| Teriflunomide HMR1726 | Teriflunomide HMR1726 | Sanofi | marketed | Dihydroorotate dehydrogenase inhibitor; immunosuppressant | Dihydroorotate dehydrogenase (DHODH) | |
| Leflunomide 10 milligram (MG) | Leflunomide 10 milligram (MG) | P. Verschueren | marketed | DHODH inhibitor; disease-modifying antirheumatic drug (DMARD) | Dihydroorotate dehydrogenase (DHODH) | |
| FLUNIXIN | FLUNIXIN | marketed | Dihydroorotate dehydrogenase (quinone), mitochondrial | |||
| Leflunomide plus Methotrexate | Leflunomide plus Methotrexate | Bangladesh Medical University | marketed | Disease-modifying antirheumatic drug (DMARD) combination | Dihydroorotate dehydrogenase (leflunomide); Dihydrofolate reductase (methotrexate) | |
| Leflunomide(LEF) | Leflunomide(LEF) | Nanjing Children's Hospital | marketed | Immunosuppressant; DHODH inhibitor | Dihydroorotate dehydrogenase (DHODH) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Pyrimidine synthesis inhibitor class)
- Beijing Biohealthcare Biotechnology Co.,Ltd · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Gimeracil and Oteracil Porassium Capsules — Competitive Intelligence Brief. https://druglandscape.com/ci/gimeracil-and-oteracil-porassium-capsules. Accessed 2026-05-18.
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