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Gemigliptin/Glimepiride combination — Competitive Intelligence Brief
phase 3
DPP-4 inhibitor + sulfonylurea combination
DPP-4 (dipeptidyl peptidase-4) and sulfonylurea receptor (SUR1)
Diabetes
Small molecule
Live · refreshed every 30 min
Target snapshot
Gemigliptin/Glimepiride combination (Gemigliptin/Glimepiride combination) — LG Life Sciences. Gemigliptin inhibits dipeptidyl peptidase-4 (DPP-4) to increase incretin levels and insulin secretion, while glimepiride stimulates pancreatic beta cells to release insulin directly.
Comparator set (2 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Gemigliptin/Glimepiride combination TARGET | Gemigliptin/Glimepiride combination | LG Life Sciences | phase 3 | DPP-4 inhibitor + sulfonylurea combination | DPP-4 (dipeptidyl peptidase-4) and sulfonylurea receptor (SUR1) | |
| Teneligliptin + Sulfonylurea | Teneligliptin + Sulfonylurea | Tanabe Pharma Corporation | phase 3 | DPP-4 inhibitor + Sulfonylurea combination | DPP-4 enzyme; ATP-sensitive potassium channels on pancreatic beta cells | |
| Alogliptin and glyburide | Alogliptin and glyburide | Takeda | phase 3 | DPP-4 inhibitor + sulfonylurea combination | DPP-4 (dipeptidyl peptidase-4) and sulfonylurea receptor (SUR1) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (DPP-4 inhibitor + sulfonylurea combination class)
- LG Life Sciences · 1 drug in this class
- Takeda · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Gemigliptin/Glimepiride combination — Competitive Intelligence Brief. https://druglandscape.com/ci/gemigliptin-glimepiride-combination. Accessed 2026-06-10.
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