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Fondaparinux Sodium (Arixtra) — Competitive Intelligence Brief
marketed
Factor Xa inhibitor
Factor Xa
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Fondaparinux Sodium (Arixtra) (Fondaparinux Sodium (Arixtra)) — Paul Di Cesare,MD. Fondaparinux selectively inhibits Factor Xa, a key enzyme in the coagulation cascade, preventing thrombin generation and blood clot formation.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Fondaparinux Sodium (Arixtra) TARGET | Fondaparinux Sodium (Arixtra) | Paul Di Cesare,MD | marketed | Factor Xa inhibitor | Factor Xa | |
| Hympavzi | MARSTACIMAB | Pfizer Inc | marketed | Monoclonal Antibody | Factor Xa | 2025-01-01 |
| Eliquis | apixaban | Bristol-Myers Squibb | marketed | Factor Xa inhibitor | Factor Xa (FXa) | 2012-01-01 |
| Xarelto | rivaroxaban | Johnson & Johnson | marketed | Direct Factor Xa Inhibitor | Factor Xa (FXa) | 2011-01-01 |
| Heparin Sodium In Plastic Container | Heparin Sodium | Fresenius Kabi | marketed | Anti-coagulant | Antithrombin III, Factor Xa, Factor IIa | 1939-01-01 |
| Heparin administration | Heparin administration | Anemia Working Group Romania | marketed | Anticoagulant | Antithrombin III (indirect); Thrombin and Factor Xa (downstream targets) | |
| Intermediate dose dalteparin | Intermediate dose dalteparin | Academisch Medisch Centrum - Universiteit van Amsterdam (AMC-UvA) | marketed | Low-molecular-weight heparin (LMWH) | Antithrombin III (indirect); Factor Xa and Thrombin (downstream targets) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Factor Xa inhibitor class)
- GlaxoSmithKline · 4 drugs in this class
- Bayer · 2 drugs in this class
- China National Center for Cardiovascular Diseases · 1 drug in this class
- Hoffmann-La Roche · 1 drug in this class
- Kim, Seok Jin · 1 drug in this class
- NYU Langone Health · 1 drug in this class
- Paul Di Cesare,MD · 1 drug in this class
- Pfizer · 1 drug in this class
- Queen Mary University of London · 1 drug in this class
- Queen's University · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Fondaparinux Sodium (Arixtra) — Competitive Intelligence Brief. https://druglandscape.com/ci/fondaparinux-sodium-arixtra. Accessed 2026-05-17.
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