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Fluzoparib; Apatinib — Competitive Intelligence Brief
phase 3
PARP inhibitor + tyrosine kinase inhibitor (combination therapy)
PARP1/PARP2; VEGFR2
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Fluzoparib; Apatinib (Fluzoparib; Apatinib) — Jiangsu HengRui Medicine Co., Ltd.. Fluzoparib is a PARP inhibitor that blocks DNA repair, while apatinib is a tyrosine kinase inhibitor targeting VEGFR2, together enhancing anti-tumor effects through synthetic lethality and anti-angiogenesis.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Fluzoparib; Apatinib TARGET | Fluzoparib; Apatinib | Jiangsu HengRui Medicine Co., Ltd. | phase 3 | PARP inhibitor + tyrosine kinase inhibitor (combination therapy) | PARP1/PARP2; VEGFR2 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (PARP inhibitor + tyrosine kinase inhibitor (combination therapy) class)
- Jiangsu HengRui Medicine Co., Ltd. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Fluzoparib; Apatinib — Competitive Intelligence Brief. https://druglandscape.com/ci/fluzoparib-apatinib. Accessed 2026-06-10.
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