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Ezetimibe/Rosuvastatin — Competitive Intelligence Brief
marketed
Cholesterol absorption inhibitor + HMG-CoA reductase inhibitor (statin combination)
NPC1L1 transporter (ezetimibe); HMG-CoA reductase (rosuvastatin)
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Ezetimibe/Rosuvastatin (Ezetimibe/Rosuvastatin) — Addpharma Inc.. This combination reduces cholesterol by blocking intestinal cholesterol absorption (ezetimibe) and inhibiting HMG-CoA reductase to decrease hepatic cholesterol synthesis (rosuvastatin).
Comparator set (1 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Ezetimibe/Rosuvastatin TARGET | Ezetimibe/Rosuvastatin | Addpharma Inc. | marketed | Cholesterol absorption inhibitor + HMG-CoA reductase inhibitor (statin combination) | NPC1L1 transporter (ezetimibe); HMG-CoA reductase (rosuvastatin) | |
| Ezetimibe + Atorvastatin | Ezetimibe + Atorvastatin | Organon and Co | marketed | Cholesterol absorption inhibitor + HMG-CoA reductase inhibitor (statin combination) | NPC1L1 (ezetimibe); HMG-CoA reductase (atorvastatin) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Cholesterol absorption inhibitor + HMG-CoA reductase inhibitor (statin combination) class)
- Addpharma Inc. · 1 drug in this class
- Organon and Co · 1 drug in this class
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- Ezetimibe/Rosuvastatin CI watch — RSS
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Cite this brief
Drug Landscape (2026). Ezetimibe/Rosuvastatin — Competitive Intelligence Brief. https://druglandscape.com/ci/ezetimibe-rosuvastatin. Accessed 2026-06-10.
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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing