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Dexbenzetimide — Competitive Intelligence Brief
phase 2
dexetimide
Muscarinic acetylcholine receptor M2
Neuroscience
Small molecule
Live · refreshed every 30 min
Target snapshot
Dexbenzetimide (DEXETIMIDE). Dexbenzetimide works by blocking the M2 muscarinic acetylcholine receptor, which helps to regulate muscle contractions and other bodily functions.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Dexbenzetimide TARGET | DEXETIMIDE | phase 2 | dexetimide | Muscarinic acetylcholine receptor M2 | ||
| Toviaz | FESOTERODINE | Pfizer | marketed | fesoterodine | Muscarinic acetylcholine receptor M2 | 2008-01-01 |
| Toviaz | Fesoterodine Fumarate | Pfizer | marketed | fesoterodine | Muscarinic acetylcholine receptor M2 | 2008-01-01 |
| HEXOCYCLIUM | HEXOCYCLIUM | AbbVie | marketed | hexocyclium | Muscarinic acetylcholine receptor M1, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M3 | 1982-01-01 |
| Syncurine | DECAMETHONIUM | marketed | decamethonium | Acetylcholinesterase, Histamine H3 receptor, Muscarinic acetylcholine receptor M2 | 1975-01-01 | |
| Cantil | MEPENZOLATE | Sanofi | marketed | Anticholinergic | Muscarinic acetylcholine receptor M2 | 1956-01-01 |
| Kemadrine | PROCYCLIDINE | marketed | Muscarinic acetylcholine receptor M1, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M3 | 1955-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
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Sponsor landscape (dexetimide class)
- · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Dexbenzetimide — Competitive Intelligence Brief. https://druglandscape.com/ci/dexetimide. Accessed 2026-06-10.
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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing