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Darolutamide Oral Tablet — Competitive Intelligence Brief
marketed
Androgen receptor antagonist
Androgen receptor (AR)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Darolutamide Oral Tablet (Darolutamide Oral Tablet) — Santa Chiara Hospital. Darolutamide is an androgen receptor antagonist that blocks the binding of androgens to the androgen receptor, inhibiting androgen-driven prostate cancer cell growth.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Darolutamide Oral Tablet TARGET | Darolutamide Oral Tablet | Santa Chiara Hospital | marketed | Androgen receptor antagonist | Androgen receptor (AR) | |
| Maximum androgen blockade | Maximum androgen blockade | Wonju Severance Christian Hospital | marketed | Androgen receptor antagonist combination therapy | Androgen receptor; testosterone synthesis pathway | |
| Zoladex and Casodex | Zoladex and Casodex | AstraZeneca | marketed | GnRH agonist (Zoladex) and androgen receptor antagonist (Casodex) | GnRH receptor (Zoladex); androgen receptor (Casodex) | |
| ODM-201 Tablet A | ODM-201 Tablet A | Orion Corporation, Orion Pharma | marketed | Androgen receptor antagonist | Androgen receptor (AR) | |
| Apalutamide Oral Tablet | Apalutamide Oral Tablet | Santa Chiara Hospital | phase 3 | Androgen receptor antagonist | Androgen receptor (AR) | |
| Abiraterone Acetate or Enzalutamide | Abiraterone Acetate or Enzalutamide | National Cancer Institute, Naples | phase 3 | Androgen synthesis inhibitor (abiraterone) / Androgen receptor antagonist (enzalutamide) | CYP17A1 (abiraterone) / Androgen receptor (enzalutamide) | |
| Darolutamide (BAY 1841788) | Darolutamide (BAY 1841788) | Canadian Cancer Trials Group | phase 3 | Non-steroidal androgen receptor antagonist | Androgen receptor (AR) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Androgen receptor antagonist class)
- Santa Chiara Hospital · 2 drugs in this class
- Cassiopea SpA · 2 drugs in this class
- The First Affiliated Hospital with Nanjing Medical University · 2 drugs in this class
- Pfizer · 2 drugs in this class
- Suzhou Kintor Pharmaceutical Inc, · 1 drug in this class
- AEterna Zentaris · 1 drug in this class
- University of Sydney · 1 drug in this class
- CHU de Quebec-Universite Laval · 1 drug in this class
- Jiangsu HengRui Medicine Co., Ltd. · 1 drug in this class
- Orion Corporation, Orion Pharma · 1 drug in this class
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- Darolutamide Oral Tablet CI watch — RSS
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Cite this brief
Drug Landscape (2026). Darolutamide Oral Tablet — Competitive Intelligence Brief. https://druglandscape.com/ci/darolutamide-oral-tablet. Accessed 2026-05-16.
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