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Conventional NSAA — Competitive Intelligence Brief
phase 3
Androgen receptor antagonist
Androgen receptor (AR)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Conventional NSAA (Conventional NSAA) — University of Sydney. Conventional NSAA (non-selective androgen antagonist) blocks androgen receptor signaling to suppress testosterone-driven prostate cancer growth.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Conventional NSAA TARGET | Conventional NSAA | University of Sydney | phase 3 | Androgen receptor antagonist | Androgen receptor (AR) | |
| Darolutamide Oral Tablet | Darolutamide Oral Tablet | Santa Chiara Hospital | marketed | Androgen receptor antagonist | Androgen receptor (AR) | |
| Zoladex and Casodex | Zoladex and Casodex | AstraZeneca | marketed | GnRH agonist (Zoladex) and androgen receptor antagonist (Casodex) | GnRH receptor (Zoladex); androgen receptor (Casodex) | |
| ODM-201 Tablet A | ODM-201 Tablet A | Orion Corporation, Orion Pharma | marketed | Androgen receptor antagonist | Androgen receptor (AR) | |
| Maximum androgen blockade | Maximum androgen blockade | Wonju Severance Christian Hospital | marketed | Androgen receptor antagonist combination therapy | Androgen receptor; testosterone synthesis pathway | |
| Abiraterone Acetate or Enzalutamide | Abiraterone Acetate or Enzalutamide | National Cancer Institute, Naples | phase 3 | Androgen synthesis inhibitor (abiraterone) / Androgen receptor antagonist (enzalutamide) | CYP17A1 (abiraterone) / Androgen receptor (enzalutamide) | |
| Proxalutamide (GT0918) | Proxalutamide (GT0918) | Suzhou Kintor Pharmaceutical Inc, | phase 3 | Androgen receptor antagonist | Androgen receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Androgen receptor antagonist class)
- Santa Chiara Hospital · 2 drugs in this class
- Cassiopea SpA · 2 drugs in this class
- The First Affiliated Hospital with Nanjing Medical University · 2 drugs in this class
- Pfizer · 2 drugs in this class
- Suzhou Kintor Pharmaceutical Inc, · 1 drug in this class
- AEterna Zentaris · 1 drug in this class
- University of Sydney · 1 drug in this class
- CHU de Quebec-Universite Laval · 1 drug in this class
- Jiangsu HengRui Medicine Co., Ltd. · 1 drug in this class
- Orion Corporation, Orion Pharma · 1 drug in this class
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- Conventional NSAA CI watch — RSS
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- Conventional NSAA alone — RSS
- Whole Androgen receptor antagonist class — RSS
Cite this brief
Drug Landscape (2026). Conventional NSAA — Competitive Intelligence Brief. https://druglandscape.com/ci/conventional-nsaa. Accessed 2026-05-13.
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