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Vaprisol In 5% Dextrose In Plastic Container — Competitive Intelligence Brief
marketed
Vasopressin Receptor Antagonist
Vasopressin V2 receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Vaprisol In 5% Dextrose In Plastic Container (CONIVAPTAN) — Cumberland.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Vaprisol In 5% Dextrose In Plastic Container TARGET | CONIVAPTAN | Cumberland | marketed | Vasopressin Receptor Antagonist | Vasopressin V2 receptor | 2005-01-01 |
| Samsca | TOLVAPTAN | Otsuka | marketed | Vasopressin V2 Receptor Antagonist [EPC] | Vasopressin V2 receptor | 2009-01-01 |
| Physulime | MOZAVAPTAN | Otsuka Pharmaceutical Co., Ltd. | marketed | mozavaptan | Vasopressin V2 receptor | 2006-01-01 |
| tolvaptan+torasemide | tolvaptan+torasemide | Shanghai Chest Hospital | marketed | Combination diuretic (vasopressin V2 receptor antagonist + loop diuretic) | Vasopressin V2 receptor (tolvaptan); Na-K-Cl cotransporter (torasemide) | |
| OPC-41061 (Tolvaptan) | OPC-41061 (Tolvaptan) | Otsuka Pharmaceutical Co., Ltd. | phase 3 | Vasopressin V2 receptor antagonist | Vasopressin V2 receptor | |
| Tolvaptan Oral Tablet | Tolvaptan Oral Tablet | Otsuka Pharmaceutical Co., Ltd. | phase 3 | Vasopressin V2-receptor antagonist (vaptans) | Vasopressin V2 receptor | |
| OPC-41061 | OPC-41061 | Otsuka Pharmaceutical Co., Ltd. | phase 3 | Vasopressin V2 receptor antagonist (vaptан) | Vasopressin V2 receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Vasopressin Receptor Antagonist class)
- Cumberland · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Vaprisol In 5% Dextrose In Plastic Container — Competitive Intelligence Brief. https://druglandscape.com/ci/conivaptan. Accessed 2026-05-13.
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