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Cycloprolol — Competitive Intelligence Brief
phase 2
cicloprolol
Beta-1 adrenergic receptor, Beta-2 adrenergic receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Cycloprolol (CICLOPROLOL). Cycloprolol works by blocking the beta-1 adrenergic receptor, which reduces the heart's workload and slows heart rate.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Cycloprolol TARGET | CICLOPROLOL | phase 2 | cicloprolol | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor | ||
| ProAir | albuterol | Generic (originally Allen & Hanburys/GSK) | marketed | SABA (Short-acting beta-2 agonist) | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Beta-2 adrenergic receptor | 1982-05-05 |
| Lopressor | metoprolol | Generic (originally Ciba-Geigy/Novartis) | marketed | Beta-1 selective blocker | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, 5-hydroxytryptamine receptor 1A | 1978-08-07 |
| Beta Blockers Carvedilol Phosphate | Beta Blockers Carvedilol Phosphate | Seoul National University Hospital | marketed | Beta blocker (non-selective, with alpha-1 blocking activity) | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| Bystolic | nebivolol | Allergan | marketed | 5-hydroxytryptamine receptor 1A, Beta-1 adrenergic receptor, Beta-2 adrenergic receptor | ||
| Serevent | Serevent | Fundacio Privada Mon Clinic Barcelona | marketed | Aldehyde oxidase, Beta-1 adrenergic receptor, Beta-2 adrenergic receptor | ||
| Carvedilol alone | Carvedilol alone | Taipei Veterans General Hospital, Taiwan | marketed | Beta-blocker with alpha-1 antagonist activity | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (cicloprolol class)
- · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Cycloprolol — Competitive Intelligence Brief. https://druglandscape.com/ci/cicloprolol. Accessed 2026-06-10.
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