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Cycloprolol — Competitive Intelligence Brief

Cycloprolol (CICLOPROLOL) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: cicloprolol. Area: Cardiovascular.

phase 2 cicloprolol Beta-1 adrenergic receptor, Beta-2 adrenergic receptor Cardiovascular Small molecule Live · refreshed every 30 min

Target snapshot

Cycloprolol (CICLOPROLOL). Cycloprolol works by blocking the beta-1 adrenergic receptor, which reduces the heart's workload and slows heart rate.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Cycloprolol TARGET CICLOPROLOL phase 2 cicloprolol Beta-1 adrenergic receptor, Beta-2 adrenergic receptor
ProAir albuterol Generic (originally Allen & Hanburys/GSK) marketed SABA (Short-acting beta-2 agonist) Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Beta-2 adrenergic receptor 1982-05-05
Lopressor metoprolol Generic (originally Ciba-Geigy/Novartis) marketed Beta-1 selective blocker Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, 5-hydroxytryptamine receptor 1A 1978-08-07
Beta Blockers Carvedilol Phosphate Beta Blockers Carvedilol Phosphate Seoul National University Hospital marketed Beta blocker (non-selective, with alpha-1 blocking activity) Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor
Bystolic nebivolol Allergan marketed 5-hydroxytryptamine receptor 1A, Beta-1 adrenergic receptor, Beta-2 adrenergic receptor
Serevent Serevent Fundacio Privada Mon Clinic Barcelona marketed Aldehyde oxidase, Beta-1 adrenergic receptor, Beta-2 adrenergic receptor
Carvedilol alone Carvedilol alone Taipei Veterans General Hospital, Taiwan marketed Beta-blocker with alpha-1 antagonist activity Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (cicloprolol class)

  1. · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Cycloprolol — Competitive Intelligence Brief. https://druglandscape.com/ci/cicloprolol. Accessed 2026-06-10.

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing