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CG5503 IR — Competitive Intelligence Brief

CG5503 IR (CG5503 IR) competitive landscape: 3 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: TRPV1 antagonist. Area: Pain Management.

phase 3 TRPV1 antagonist TRPV1 (Transient Receptor Potential Vanilloid 1) Pain Management Small molecule Live · refreshed every 30 min

Target snapshot

CG5503 IR (CG5503 IR) — Grünenthal GmbH. CG5503 is a selective inhibitor of transient receptor potential vanilloid 1 (TRPV1) that reduces pain signaling by blocking capsaicin-sensitive nociceptors.

Comparator set (3 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
CG5503 IR TARGET CG5503 IR Grünenthal GmbH phase 3 TRPV1 antagonist TRPV1 (Transient Receptor Potential Vanilloid 1)
KPI-121 Ophthalmic Suspension KPI-121 Ophthalmic Suspension Kala Pharmaceuticals, Inc. phase 3 TRPV1 antagonist / Topical anti-inflammatory TRPV1 (Transient Receptor Potential Vanilloid 1)
KPS-0373, High dose KPS-0373, High dose Kissei Pharmaceutical Co., Ltd. phase 3 TRPV1 antagonist TRPV1
TV-44749 TV-44749 Teva Branded Pharmaceutical Products R&D LLC phase 3 TRPV1 antagonist TRPV1 (Transient Receptor Potential Vanilloid 1)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (TRPV1 antagonist class)

  1. Allergan · 1 drug in this class
  2. Grünenthal GmbH · 1 drug in this class
  3. Kissei Pharmaceutical Co., Ltd. · 1 drug in this class
  4. Teva Branded Pharmaceutical Products R&D LLC · 1 drug in this class

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Cite this brief

Drug Landscape (2026). CG5503 IR — Competitive Intelligence Brief. https://druglandscape.com/ci/cg5503-ir. Accessed 2026-05-15.

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