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Burcol — Competitive Intelligence Brief
phase 2
carbutamide
Sulfonylurea receptor 1, Kir6.2
Metabolic
Small molecule
Live · refreshed every 30 min
Target snapshot
Burcol (CARBUTAMIDE). Burcol works by binding to the sulfonylurea receptor 1, Kir6.2, to stimulate insulin release from pancreatic beta cells.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Burcol TARGET | CARBUTAMIDE | phase 2 | carbutamide | Sulfonylurea receptor 1, Kir6.2 | ||
| Starlix | NATEGLINIDE | Novartis | marketed | Glinide [EPC] | Sulfonylurea receptor 1, Kir6.2 | 2000-01-01 |
| Amaryl | GLIMEPIRIDE | Sanofi | marketed | Sulfonylurea [EPC] | Sulfonylurea receptor 1, Kir6.2 | 1995-01-01 |
| Glucotrol | GLIPIZIDE | Pfizer | marketed | Sulfonylurea [EPC] | Sulfonylurea receptor 1, Kir6.2 | 1984-01-01 |
| Micronase | glibenclamide | Sanofi | marketed | Sulfonylurea | Sulfonylurea receptor 1, Kir6.2 | 1984-01-01 |
| Proglycem | DIAZOXIDE | marketed | diazoxide | Sulfonylurea receptor 1, Kir6.2 | 1973-01-01 | |
| Dymelor | ACETOHEXAMIDE | Eli Lilly | marketed | acetohexamide | Sulfonylurea receptor 1, Kir6.2 | 1964-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (carbutamide class)
- · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Burcol — Competitive Intelligence Brief. https://druglandscape.com/ci/carbutamide. Accessed 2026-06-10.
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