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Brexpiprazole +ADT — Competitive Intelligence Brief
Target snapshot
Brexpiprazole +ADT (Brexpiprazole +ADT) — Otsuka Pharmaceutical Development & Commercialization, Inc.. Brexpiprazole is an atypical antipsychotic that acts as a dopamine D2 receptor partial agonist and serotonin 5-HT1A receptor partial agonist, combined with adjunctive antidepressant therapy (ADT) to treat major depressive disorder.
Comparator set (3 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Brexpiprazole +ADT TARGET | Brexpiprazole +ADT | Otsuka Pharmaceutical Development & Commercialization, Inc. | phase 3 | Atypical antipsychotic (dopamine D2 partial agonist) | Dopamine D2 receptor, Serotonin 5-HT1A receptor | |
| Abilify MyCite® | Abilify MyCite® | Otsuka Pharmaceutical Development & Commercialization, Inc. | marketed | Atypical antipsychotic with digital adherence monitoring | Dopamine D2 receptor, serotonin 5-HT1A receptor | |
| Adjunct brexpiprazole | Adjunct brexpiprazole | H. Lundbeck A/S | phase 3 | Serotonin-dopamine activity modulator (SDAM) | Dopamine D2 receptor, Serotonin 5-HT1A receptor | |
| Aripiprazole (Fixed dose) | Aripiprazole (Fixed dose) | Otsuka Pharmaceutical Co., Ltd. | phase 3 | Atypical antipsychotic | Dopamine D2 receptor, Serotonin 5-HT1A receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Atypical antipsychotic (dopamine D2 partial agonist) class)
- Otsuka Pharmaceutical Development & Commercialization, Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Brexpiprazole +ADT — Competitive Intelligence Brief. https://druglandscape.com/ci/brexpiprazole-adt. Accessed 2026-06-10.
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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing