Last reviewed · How we verify
BL - 1020 — Competitive Intelligence Brief
phase 2
Vasopressin V2 receptor antagonist
V2 receptor
Nephrology
Small molecule
Live · refreshed every 30 min
Target snapshot
BL - 1020 (BL - 1020) — BioLineRx, Ltd.. BL-1020 is a vasopressin V2 receptor antagonist.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| BL - 1020 TARGET | BL - 1020 | BioLineRx, Ltd. | phase 2 | Vasopressin V2 receptor antagonist | V2 receptor | |
| Samsca | TOLVAPTAN | Otsuka | marketed | Vasopressin V2 Receptor Antagonist [EPC] | Vasopressin V2 receptor | 2009-01-01 |
| Physulime | MOZAVAPTAN | Otsuka Pharmaceutical Co., Ltd. | marketed | mozavaptan | Vasopressin V2 receptor | 2006-01-01 |
| Vaprisol In 5% Dextrose In Plastic Container | CONIVAPTAN | Cumberland | marketed | Vasopressin Receptor Antagonist | Vasopressin V2 receptor | 2005-01-01 |
| tolvaptan+torasemide | tolvaptan+torasemide | Shanghai Chest Hospital | marketed | Combination diuretic (vasopressin V2 receptor antagonist + loop diuretic) | Vasopressin V2 receptor (tolvaptan); Na-K-Cl cotransporter (torasemide) | |
| Tolvaptan Tablets | Tolvaptan Tablets | Institute of Liver and Biliary Sciences, India | phase 3 | Vasopressin receptor antagonist | V2 receptor | |
| Vasopressin administration | Vasopressin administration | Assistance Publique Hopitaux De Marseille | phase 3 | Vasopressin receptor agonist | V1A and V2 receptors |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Vasopressin V2 receptor antagonist class)
- BioLineRx, Ltd. · 1 drug in this class
- Cardiovascular Clinical Sciences Inc · 1 drug in this class
- Otsuka Pharmaceutical Co., Ltd. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). BL - 1020 — Competitive Intelligence Brief. https://druglandscape.com/ci/bl-1020. Accessed 2026-05-14.
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