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bitopertin [RO4917838] level 1 — Competitive Intelligence Brief
phase 3
Glycine transporter 1 (GlyT1) inhibitor
GlyT1 (SLC6A9)
Psychiatry/Neurology
Small molecule
Live · refreshed every 30 min
Target snapshot
bitopertin [RO4917838] level 1 (bitopertin [RO4917838] level 1) — Hoffmann-La Roche. Bitopertin is a glycine transporter 1 (GlyT1) inhibitor that increases synaptic glycine levels to enhance NMDA receptor function in the brain.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| bitopertin [RO4917838] level 1 TARGET | bitopertin [RO4917838] level 1 | Hoffmann-La Roche | phase 3 | Glycine transporter 1 (GlyT1) inhibitor | GlyT1 (SLC6A9) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Glycine transporter 1 (GlyT1) inhibitor class)
- Hoffmann-La Roche · 1 drug in this class
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Cite this brief
Drug Landscape (2026). bitopertin [RO4917838] level 1 — Competitive Intelligence Brief. https://druglandscape.com/ci/bitopertin-ro4917838-level-1. Accessed 2026-05-17.
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