Last reviewed · How we verify

bitopertin [RO4917838] level 1 — Competitive Intelligence Brief

bitopertin [RO4917838] level 1 (bitopertin [RO4917838] level 1) competitive landscape: 0 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Glycine transporter 1 (GlyT1) inhibitor. Area: Psychiatry/Neurology.

phase 3 Glycine transporter 1 (GlyT1) inhibitor GlyT1 (SLC6A9) Psychiatry/Neurology Small molecule Live · refreshed every 30 min

Target snapshot

bitopertin [RO4917838] level 1 (bitopertin [RO4917838] level 1) — Hoffmann-La Roche. Bitopertin is a glycine transporter 1 (GlyT1) inhibitor that increases synaptic glycine levels to enhance NMDA receptor function in the brain.

Comparator set

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
bitopertin [RO4917838] level 1 TARGET bitopertin [RO4917838] level 1 Hoffmann-La Roche phase 3 Glycine transporter 1 (GlyT1) inhibitor GlyT1 (SLC6A9)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Glycine transporter 1 (GlyT1) inhibitor class)

  1. Hoffmann-La Roche · 1 drug in this class

Subscribe to ongoing alerts

Push every new event for this competitive set into your RSS reader, IFTTT/Zapier workflow, or email digest:

Cite this brief

Drug Landscape (2026). bitopertin [RO4917838] level 1 — Competitive Intelligence Brief. https://druglandscape.com/ci/bitopertin-ro4917838-level-1. Accessed 2026-05-17.

Build your own brief

Pick any drug + add comparators: