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Saphris — Competitive Intelligence Brief
marketed
Atypical Antipsychotic [EPC]
5-hydroxytryptamine receptor 2C
Neuroscience
Small molecule
Live · refreshed every 30 min
Target snapshot
Saphris (ASENAPINE) — Hisamitsu. Saphris works by blocking the action of serotonin at the 5-hydroxytryptamine receptor 2C.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Saphris TARGET | ASENAPINE | Hisamitsu | marketed | Atypical Antipsychotic [EPC] | 5-hydroxytryptamine receptor 2C | 2009-01-01 |
| Belviq | LORCASERIN | Eisai | marketed | Serotonin-2c Receptor Agonist | 5-hydroxytryptamine receptor 2C | 2012-01-01 |
| Remeron | mirtazapine | Generic (originally Organon/MSD) | marketed | NaSSA (Noradrenergic and specific serotonergic antidepressant) | 5-hydroxytryptamine receptor 1A, 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2C | 1996-06-14 |
| Zerdol | SERTINDOLE | H. Lundbeck A/S | marketed | sertindole | 5-hydroxytryptamine receptor 2C | 1996-01-01 |
| Effexor | venlafaxine | Generic (originally Wyeth/Pfizer) | marketed | SNRI (Serotonin-norepinephrine reuptake inhibitor) | 5-hydroxytryptamine receptor 6, 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2C | 1993-12-28 |
| Amoxil | amoxicillin | Generic (originally Beecham/GSK) | marketed | Aminopenicillin (Beta-lactam antibiotic) | 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2B, 5-hydroxytryptamine receptor 2C | 1972-01-01 |
| Amoxicilli | Amoxicilli | Shandong Luoxin Pharmaceutical Group Stock Co., Ltd. | marketed | 5-hydroxytryptamine receptor 2A, 5-hydroxytryptamine receptor 2B, 5-hydroxytryptamine receptor 2C |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
- — Amoxil · 8778924 · Compound · US
- — Amoxil · 8357394 · Formulation · US
- — Amoxil · 8299052 · Method of Use · US
Sponsor landscape (Atypical Antipsychotic [EPC] class)
- · 2 drugs in this class
- AbbVie · 1 drug in this class
- Alkermes Inc · 1 drug in this class
- Eli Lilly · 1 drug in this class
- Hisamitsu · 1 drug in this class
- Intra-Cellular · 1 drug in this class
- Jazz Pharmaceuticals · 1 drug in this class
- Johnson & Johnson (Janssen) · 1 drug in this class
- Otsuka · 1 drug in this class
- Vanda Pharms Inc · 1 drug in this class
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- Whole Atypical Antipsychotic [EPC] class — RSS
Cite this brief
Drug Landscape (2026). Saphris — Competitive Intelligence Brief. https://druglandscape.com/ci/asenapine. Accessed 2026-05-13.
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