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aripiprazole long acting injectable formulation — Competitive Intelligence Brief
marketed
Atypical antipsychotic (dopamine partial agonist)
Dopamine D2 receptor, Dopamine D3 receptor
Psychiatry / Neurology
Small molecule
Live · refreshed every 30 min
Target snapshot
aripiprazole long acting injectable formulation (aripiprazole long acting injectable formulation) — Vanguard Research Group. Aripiprazole is a dopamine D2/D3 receptor partial agonist that modulates dopaminergic and serotonergic neurotransmission to treat psychotic and mood disorders.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| aripiprazole long acting injectable formulation TARGET | aripiprazole long acting injectable formulation | Vanguard Research Group | marketed | Atypical antipsychotic (dopamine partial agonist) | Dopamine D2 receptor, Dopamine D3 receptor | |
| ropinirole CR-RLS | ropinirole CR-RLS | GlaxoSmithKline | marketed | Dopamine D2/D3 receptor agonist | Dopamine D2 receptor, Dopamine D3 receptor | |
| [11C]raclopride | [11C]raclopride | New York State Psychiatric Institute | marketed | Dopamine D2/D3 receptor antagonist (PET imaging agent) | Dopamine D2 receptor, Dopamine D3 receptor | |
| IM aripiprazole once monthly | IM aripiprazole once monthly | University of Utah | marketed | Atypical antipsychotic | Dopamine D2 receptor, Dopamine D3 receptor | |
| Raclopride C11 | Raclopride C11 | University of North Carolina, Chapel Hill | marketed | Dopamine D2/D3 receptor antagonist (PET imaging agent) | Dopamine D2 receptor, Dopamine D3 receptor | |
| Ropinirole (Requip) | Ropinirole (Requip) | St. Luke's-Roosevelt Hospital Center | marketed | Dopamine D2/D3 receptor agonist | Dopamine D2 receptor, Dopamine D3 receptor | |
| Amisulpride add-on | Amisulpride add-on | National Health Research Institutes, Taiwan | marketed | Atypical antipsychotic | Dopamine D2 receptor, Dopamine D3 receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Atypical antipsychotic (dopamine partial agonist) class)
- Vanguard Research Group · 1 drug in this class
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Cite this brief
Drug Landscape (2026). aripiprazole long acting injectable formulation — Competitive Intelligence Brief. https://druglandscape.com/ci/aripiprazole-long-acting-injectable-formulation. Accessed 2026-05-14.
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