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APL-130277 — Competitive Intelligence Brief
phase 3
Dopamine agonist
Dopamine receptors (D1, D2)
Neurology
Small molecule
Live · refreshed every 30 min
Target snapshot
APL-130277 (APL-130277) — Sumitomo Pharma America, Inc.. APL-130277 is a subcutaneous apomorphine formulation that acts as a dopamine agonist to provide rapid symptom relief in Parkinson's disease.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| APL-130277 TARGET | APL-130277 | Sumitomo Pharma America, Inc. | phase 3 | Dopamine agonist | Dopamine receptors (D1, D2) | |
| Neupro | ROTIGOTINE | UCB | marketed | Nonergot Dopamine Agonist [EPC] | dopamine receptors | 2007-01-01 |
| DC | DC | Gary Archer Ph.D. | marketed | dopamine agonist | dopamine receptor | |
| Rotigotine transdermal patch | Rotigotine transdermal patch | UCB BIOSCIENCES GmbH | marketed | Non-ergot dopamine agonist | Dopamine receptors (D1, D2, D3, D4, D5) | |
| ROP+L-Dopa | ROP+L-Dopa | GlaxoSmithKline | marketed | Dopamine agonist + Levodopa combination | Dopamine receptors (D2/D3); Dopamine pathway | |
| DAM | DAM | Beijing Bozhiyin T&S Co., Ltd. | marketed | Dopamine agonist | Dopamine receptor | |
| amantadine sulfate | amantadine sulfate | Jee-Young Lee | marketed | Antiviral / Dopamine agonist | Influenza A M2 ion channel; dopamine system (mechanism not fully elucidated) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Dopamine agonist class)
- Sumitomo Pharma America, Inc. · 2 drugs in this class
- University Hospital, Toulouse · 2 drugs in this class
- Rennes University Hospital · 2 drugs in this class
- Britannia Pharmaceuticals Ltd. · 1 drug in this class
- Desitin Arzneimittel GmbH · 1 drug in this class
- GlaxoSmithKline · 1 drug in this class
- Intec Pharma Ltd. · 1 drug in this class
- Leiden University Medical Center · 1 drug in this class
- Ludwig-Maximilians - University of Munich · 1 drug in this class
- Massachusetts General Hospital · 1 drug in this class
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Cite this brief
Drug Landscape (2026). APL-130277 — Competitive Intelligence Brief. https://druglandscape.com/ci/apl-130277. Accessed 2026-05-14.
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